KDM5A-IN-1 |
| Catalog No.GC32842 |
KDM5A-IN-1 es un potente inhibidor biodisponible por vÍa oral de panhistona lisina desmetilasas 5 (KDM5) con IC50 de 45 nM, 56 nM y 55 nM para KDM5A, KDM5B y KDM5C, respectivamente, y con un valor EC50 de 960 nM para PC9 H3K4Me3. KDM5A-IN-1 es significativamente menos potente frente a otras enzimas KDM5B (1A, 2B, 3B, 4C, 6A, 7B).
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 1905481-36-8
Sample solution is provided at 25 µL, 10mM.
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KDM5A-IN-1 is an inhibitor histone demethylases. Target: Histone Demethylase
[1]. Kwong Wah LAI, et al. Pyrrolidine amide compounds as histone demethylase inhibitors. PCT Int. Appl. (2016), WO 2016057924 A1 20160414.
Average Rating: 5 (Based on Reviews and 13 reference(s) in Google Scholar.)
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