GPCR/G protein
Research Areas
- Neuropeptide FF/AF Receptors(54)
- Neuropeptide S Receptor(3)
- GPBA Receptor(5)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- Formyl Peptide Receptors(11)
- 5-HT Receptor(433)
- Acetylcholine(28)
- Adenosine Deaminase(10)
- Adenosine Receptor(143)
- Adenosine Kinase(5)
- Adiponectin Receptor(3)
- Adrenergic Receptor(452)
- Adrenergic Transporters(5)
- Apelin Receptor(9)
- Angiotensin Receptor(118)
- Bombesin Receptors(26)
- Bradykinin Receptors(30)
- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(121)
- Calcimimetic Agent(2)
- CaSR(28)
- CCK1 Receptors(7)
- CCK2 Receptors(7)
- CCR(98)
- Chemokine Receptors(23)
- CRF1 Receptors(10)
- CRF2 Receptors(3)
- CXCR(109)
- CysLT1 receptor(1)
- Endothelin Receptor(54)
- EP1 Receptor(2)
- EP4 Receptor(2)
- ERRγ(1)
- ETA Receptors(5)
- ETB Receptors(5)
- Free Fatty Acid Receptors(16)
- Galanin Receptors(11)
- Ghrelin Receptors(11)
- GHSR(20)
- GIP Receptor(5)
- Glucagon Receptor(54)
- Glucocorticoid Receptor(103)
- GLUT1(1)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(12)
- GPR109A(4)
- GPR119(11)
- GPR120(9)
- GPR35(10)
- GPR44(1)
- GPR55(11)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(57)
- LPA Receptor(12)
- LPL Receptor(64)
- LTD4 Receptor(1)
- mGluR (127)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(62)
- Melatonin Receptors(23)
- Motilin Receptor(7)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(26)
- NK2 Receptors(7)
- NK3 Receptor(5)
- NOP Receptor(20)
- NPY Receptors(26)
- Orexin(3)
- Orphan 7-TM Receptors(6)
- OX Receptor(58)
- Oxytocin Receptors(22)
- P2Y Receptor(66)
- PACAP Receptors(7)
- PAF Receptors(7)
- Peptide Receptors(14)
- PGD2 Receptor(1)
- Prostaglandin Receptor(179)
- Prostanoid Receptors(25)
- Protease-Activated Receptors(9)
- RGS(2)
- S1P receptor(8)
- Secretin Receptors(1)
- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(47)
- Sigma Receptor(62)
- Vasopressin Receptor(34)
- 17,20-lyase(4)
- Ras(182)
- Urotensin-II Receptor(10)
- VIP Receptors(6)
- EBI2/GPR183(7)
- TSH Receptor(12)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(20)
- GPR84(11)
- Neuromedin U Receptors(2)
- Kisspeptin Receptor(8)
- CRFR(29)
- RGS Protein(5)
- Urotensin Receptor(7)
- Cholecystokinin Receptor(29)
- GPR139(4)
- mAChR(201)
- MCHR1 (GPR24)(17)
- Neurokinin Receptor(78)
- cGMP(27)
- GRK(5)
- GPR88(3)
- Amylin Receptor(9)
- Arrestin(11)
- Mas-related G-protein-coupled Receptor (MRGPR)(10)
- GCGR(13)
- GLP Receptor(27)
- Succinate Receptor 1(2)
- PTHR(3)
- Protease Activated Receptor (PAR)(6)
- Free Fatty Acid Receptor(5)
- Formyl Peptide Receptor (FPR)(7)
- Hydroxycarboxylic Acid Receptor (HCAR)(2)
- RXFP Receptor(3)
- Adhesion G Protein-coupled Receptors (AGPCRs)(1)
- Taste Receptor(1)
- GPR52(1)
Products Related to GPCR/G protein(3744)
- GC84659Anti-TSHR Antibody (K1-70)Purity: >98.00%
Anti-TSHR Antibody (K1-70) is an anti- TSHR monoclonal antibody.
- GC84688Gastrin I (1-14), human TFAPurity: >99.00%
Gastrin I (1-14), human TFA is 1-14 fragment of human gastrin I peptide.
- GC84692BIIE-0246 hydrochloridePurity: >99.00%
BIIE-0246 hydrochloride (AR-H 053591 hydrochloride) is a potent and selective NPY2R ( neuropeptide Y receptor 2) antagonist with an IC 50 value of 15 nM for rat [ 125 I]PYY 3-36.
- GC846935-HT2C agonist-3CAS: 2104810-18-4Purity: >99.50%
5-HT2C agonist-3 ((+)-19) is a selective 5-HT2C agonist ( EC 50: 24 nM, K i: 78 nM).
- GC84698Zinterol hydrochlorideCAS: 38241-28-0Purity: >99.50%
Zinterol hydrochloride (MJ 9184 hydrochloride) is a potent and selective β2-adrenoceptor agonist [1] . Zinterol hydrochloride increases I Ca in a concentration-dependent manner with an EC 50 of 2.2 nM [2] . Zinterol hydrochloride induces ventricular arrhythmias in conscious heart failure rabbits [3] .
- GC84723(+)-SotalolCAS: 30236-32-9Purity: >99.50%
(+)-Sotalol ((S)-Sotalol) is the S-isomer of Sotalol.
- GC84752Calhex 231 hydrochlorideCAS: 2387505-78-2Purity: >99.00%
Calhex 231 hydrochloride is a potent negative allosteric modulator that blocks (IC 50 = 0.39 μM) increases in [ 3 H]inositol phosphates elicited by activating the human wild-type CaSR transiently Ca 2+ -sensing receptor.
- GC84780Glucagon-like peptide 1 (1-37), human TFAPurity: >99.50%
Glucagon-like peptide 1 (1-37), human (TFA) is a highly potent agonist of the GLP-1 receptor.
- GC84823α-Helical CRF(9-41) TFAPurity: >99.50%
α-Helical CRF(9-41) TFA is a competitive CRF2 receptor antagonist with K B of ~100 nM.
- GC84826Urocortin III, mouse TFAPurity: >98.00%
Urocortin III, mouse TFA is a corticotropin-releasing factor ( CRF )-related peptide.
- GN10659TheophyllineCAS: 58-55-9Purity: >99.50%
Theophylline is a nonspecific phosphodiesterase (PDE) inhibitor, adenosine receptor antagonist, and histone deacetylase (HDAC) activator.
- GA20063(D-Ala2)-GIP (human)CAS: 444073-04-5Purity: >95.50%
(D-Ala2)-GIP (human) is an analog of glucose-dependent insulinotropic polypeptide that activates the GIP receptor (EC 50 =630pM) and is commonly used in research on type 2 diabetes treatment.
- GA20155(D-Pro⁷)-Angiotensin I/II (1-7)CAS: 586962-44-9Purity: 98.68%
(D-Pro⁷)-Angiotensin I/II (1-7) is a peptide antagonist of the Mas receptor, engineered by replacing the C-terminal Pro⁷ of Angiotensin-(1-7) with a D-proline.
- GA20195(Gly¹,Ser³·²²,Gln⁴·³⁴,Thr⁶,Arg¹⁹,Tyr²¹,Ala²³·³¹,Aib³²)-Pancreatic Polypeptide (human)CAS: 313988-89-5Purity: >98.00%
(Gly¹,Ser³.²²,Gln⁴.³⁴,Thr⁶,Arg¹⁹,Tyr²¹,Ala²³.³¹,Aib³²)-Pancreatic Polypeptide (human) هو ناهض مستقبلات الببتيد العصبي Y5 القوي والانتقائي مع IC50 من 0.24 نانومتر للارتباط بمستقبل hY5.
- GA20221(Hyp³)-BradykininCAS: 37642-65-2Purity: >98.00%
(Hyp³ ؛) - براديكينين ، هرمون الببتيد الذي يحدث بشكل طبيعي ، هو ناهض مستقبلات البراديكينين.
- GA20228(Leu¹⁵)-Gastrin I (human)CAS: 39024-57-2Purity: >98.00%
يُمثّل (Leu¹⁵)-Gastrin I (human) مشتقاً ببتيدياً لهرمون الغاسترين I، ويمتاز بقدرته على الارتباط المتشابك بالأغشية البلازمية أو الخلايا الجدارية السليمة.
- GA20229(Leu³¹,Pro³⁴)-Neuropeptide Y (human, rat)CAS: 132699-73-1Purity: >98.00%
(Leu³؛ ¹؛، Pro³؛ ⁴) -Neuropeptide Y (الإنسان ، الجرذ) هو ناهض مستقبلات الببتيد العصبي Y1 المحدد.
- GA20291(Sar¹)-Angiotensin IICAS: 51833-69-3Purity: >98.00%
(Sar¹ ؛) - أنجيوتنسين 2 ، نظير أنجيوتنسين 2 ، هو ناهض محدد لمستقبلات الأنجيوتنسين AT1.
- GA20643Ac-Pro-Gly-Pro-OHCAS: 292171-04-1Purity: >98.00%
Ac-Pro-Gly-Pro-OH is an endogenous degradation product of extracellular collagen and acts as a CXCR2 agonist.
- GA20760Angiotensin A (1-7)CAS: 1176306-10-7Purity: >98.50%
أنجيوتنسين أ (1-7) ، عضو في نظام الرينين-أنجيوتنسين (RAS) ، ببتيد فعال في الأوعية ، عبارة عن ليجند داخلي من مستقبلات البروتين G المرتبط بـ MrgD.
- GA20807Big Endothelin-1 (1-38), humanCAS: 120796-97-6Purity: >98.00%
Big Endothelin-1 (1-38) ، الإنسان هو مقدمة من endothelin-1.
| Catalog No. | Product Name | CAS No. | Purity | Structure |
|---|---|---|---|---|
| GC84659 | Anti-TSHR Antibody (K1-70) | - | >98.00% | |
Anti-TSHR Antibody (K1-70) is an anti- TSHR monoclonal antibody. | ||||
| GC84676 | NI-0701 | - | >99.50% | |
NI-0701 is a humanized antibody expressed in CHO cells that targets CCL5/RANTES. | ||||
| GC84688 | Gastrin I (1-14), human TFA | - | >99.00% | |
Gastrin I (1-14), human TFA is 1-14 fragment of human gastrin I peptide. | ||||
| GC84692 | BIIE-0246 hydrochloride | - | >99.00% | |
BIIE-0246 hydrochloride (AR-H 053591 hydrochloride) is a potent and selective NPY2R ( neuropeptide Y receptor 2) antagonist with an IC 50 value of 15 nM for rat [ 125 I]PYY 3-36. | ||||
| GC84693 | 5-HT2C agonist-3 | 2104810-18-4 | >99.50% | |
5-HT2C agonist-3 ((+)-19) is a selective 5-HT2C agonist ( EC 50: 24 nM, K i: 78 nM). | ||||
| GC84698 | Zinterol hydrochloride | 38241-28-0 | >99.50% | |
Zinterol hydrochloride (MJ 9184 hydrochloride) is a potent and selective β2-adrenoceptor agonist [1] . Zinterol hydrochloride increases I Ca in a concentration-dependent manner with an EC 50 of 2.2 nM [2] . Zinterol hydrochloride induces ventricular arrhythmias in conscious heart failure rabbits [3] . | ||||
| GC84723 | (+)-Sotalol | 30236-32-9 | >99.50% | |
(+)-Sotalol ((S)-Sotalol) is the S-isomer of Sotalol. | ||||
| GC84752 | Calhex 231 hydrochloride | 2387505-78-2 | >99.00% | |
Calhex 231 hydrochloride is a potent negative allosteric modulator that blocks (IC 50 = 0.39 μM) increases in [ 3 H]inositol phosphates elicited by activating the human wild-type CaSR transiently Ca 2+ -sensing receptor. | ||||
| GC84768 | (-)-ZK 216348 | - | >99.50% | |
(-)-ZK 216348 is the enantiomer of (+)-ZK 216348. | ||||
| GC84780 | Glucagon-like peptide 1 (1-37), human TFA | - | >99.50% | |
Glucagon-like peptide 1 (1-37), human (TFA) is a highly potent agonist of the GLP-1 receptor. | ||||
| GC84787 | vMIP-II (1-21) TFA | - | - | |
vMIP-II (1-21) (NT21MP) TFA is an inhibitor of CXCR4. | ||||
| GC84823 | α-Helical CRF(9-41) TFA | - | >99.50% | |
α-Helical CRF(9-41) TFA is a competitive CRF2 receptor antagonist with K B of ~100 nM. | ||||
| GC84826 | Urocortin III, mouse TFA | - | >98.00% | |
Urocortin III, mouse TFA is a corticotropin-releasing factor ( CRF )-related peptide. | ||||
| GN10659 | Theophylline | 58-55-9 | >99.50% | |
Theophylline is a nonspecific phosphodiesterase (PDE) inhibitor, adenosine receptor antagonist, and histone deacetylase (HDAC) activator. | ||||
| GA20063 | (D-Ala2)-GIP (human) | 444073-04-5 | >95.50% | |
(D-Ala2)-GIP (human) is an analog of glucose-dependent insulinotropic polypeptide that activates the GIP receptor (EC 50 =630pM) and is commonly used in research on type 2 diabetes treatment. | ||||
| GA20155 | (D-Pro⁷)-Angiotensin I/II (1-7) | 586962-44-9 | 98.68% | |
(D-Pro⁷)-Angiotensin I/II (1-7) is a peptide antagonist of the Mas receptor, engineered by replacing the C-terminal Pro⁷ of Angiotensin-(1-7) with a D-proline. | ||||
| GA20195 | (Gly¹,Ser³·²²,Gln⁴·³⁴,Thr⁶,Arg¹⁹,Tyr²¹,Ala²³·³¹,Aib³²)-Pancreatic Polypeptide (human) | 313988-89-5 | >98.00% | |
(Gly¹,Ser³.²²,Gln⁴.³⁴,Thr⁶,Arg¹⁹,Tyr²¹,Ala²³.³¹,Aib³²)-Pancreatic Polypeptide (human) هو ناهض مستقبلات الببتيد العصبي Y5 القوي والانتقائي مع IC50 من 0.24 نانومتر للارتباط بمستقبل hY5. | ||||
| GA20221 | (Hyp³)-Bradykinin | 37642-65-2 | >98.00% | |
(Hyp³ ؛) - براديكينين ، هرمون الببتيد الذي يحدث بشكل طبيعي ، هو ناهض مستقبلات البراديكينين. | ||||
| GA20228 | (Leu¹⁵)-Gastrin I (human) | 39024-57-2 | >98.00% | |
يُمثّل (Leu¹⁵)-Gastrin I (human) مشتقاً ببتيدياً لهرمون الغاسترين I، ويمتاز بقدرته على الارتباط المتشابك بالأغشية البلازمية أو الخلايا الجدارية السليمة. | ||||
| GA20229 | (Leu³¹,Pro³⁴)-Neuropeptide Y (human, rat) | 132699-73-1 | >98.00% | |
(Leu³؛ ¹؛، Pro³؛ ⁴) -Neuropeptide Y (الإنسان ، الجرذ) هو ناهض مستقبلات الببتيد العصبي Y1 المحدد. | ||||
| GA20291 | (Sar¹)-Angiotensin II | 51833-69-3 | >98.00% | |
(Sar¹ ؛) - أنجيوتنسين 2 ، نظير أنجيوتنسين 2 ، هو ناهض محدد لمستقبلات الأنجيوتنسين AT1. | ||||
| GA20643 | Ac-Pro-Gly-Pro-OH | 292171-04-1 | >98.00% | |
Ac-Pro-Gly-Pro-OH is an endogenous degradation product of extracellular collagen and acts as a CXCR2 agonist. | ||||
| GA20760 | Angiotensin A (1-7) | 1176306-10-7 | >98.50% | |
أنجيوتنسين أ (1-7) ، عضو في نظام الرينين-أنجيوتنسين (RAS) ، ببتيد فعال في الأوعية ، عبارة عن ليجند داخلي من مستقبلات البروتين G المرتبط بـ MrgD. | ||||
| GA20807 | Big Endothelin-1 (1-38), human | 120796-97-6 | >98.00% | |
Big Endothelin-1 (1-38) ، الإنسان هو مقدمة من endothelin-1. | ||||