PD-159020 |
| Catalog No.GC34031 |
PD-159020 est un antagoniste ETA/ETB non sélectif, avec des IC50 de 30 et 50 nM pour hETA et hETB, respectivement.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 177904-00-6
Sample solution is provided at 25 µL, 10mM.
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PD-159020 is a non-selective ETA/ETB antagonist, with IC50s of 30 and 50 nM for hETA and hETB, respectively.
PD-159020 demonstrates excellent inhibition of arachidonic acid release, AAR-B, with an IC50 of 0.23 μM.
[1]. Amy Mbunker, et al. 1,3-diaryl-2-carboxyindoles as potent non-peptide endothelin antagonists. Bioorganic & Medicinal Chemistry Letters. Volume 6, Issue 9, 7 May 1996, Pages 1061-1066
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