E3 ligase Ligand 1A (Synonyms: VHL ligand 2; E3 ligase Ligand 1A) |
Catalog No.GC33101 |
El ligando 1A de la ligasa E3 (ligando VHL 2) es el ligando VHL basado en (S,R,S)-AHPC que se utiliza en el reclutamiento de la proteÍna de von Hippel-Lindau (VHL). El ligando 1A de ligasa E3 se puede utilizar para sintetizar ARV-771, un degradador BET PROTAC basado en ligasa E3 de von Hippel-Landau (VHL). ARV-771 degrada potentemente la proteÍna BET en células de cÁncer de prÓstata resistente a la castraciÓn (CRPC) con un DC50 <1 nM.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 1948273-02-6
Sample solution is provided at 25 µL, 10mM.
E3 ligase Ligand 1A is a ligand of E3 ligase, used in PROTAC technology; E3 ligase Ligand 1A can be used in the research of cancer.
Average Rating: 5
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