MK-0249 |
Catalog No.GC31027 |
MK-0249 (Compuesto 1) es un antagonista del receptor de histamina H3 potente, selectivo y activo por vÍa oral, con una IC50 de 1,7 nM para H3 humano.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 862309-06-6
Sample solution is provided at 25 µL, 10mM.
MK-0249 is a potent histamine H3 receptor antagonist, with Ki of 1.7 nM for human H3.
[1]. Brioni JD, et al. Discovery of histamine H3 antagonists for the treatment of cognitive disorders and Alzheimer's disease. J Pharmacol Exp Ther. 2011 Jan;336(1):38-46.
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