>>Signaling Pathways>> Neuroscience>> Histamine Receptor>>MK-0249

MK-0249

Catalog No.GC31027

MK-0249(화합물 1)는 인간 H3에 대해 IC50이 1.7nM인 강력하고 선택적이고 경구 활성인 히스타민 H3 수용체 길항제입니다.

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MK-0249 Chemical Structure

Cas No.: 862309-06-6

Size 가격 재고 수량
1mg
US$534.00
재고 있음
5mg
US$1,057.00
재고 있음
10mg
US$1,801.00
재고 있음
20mg
US$3,171.00
재고 있음

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Sample solution is provided at 25 µL, 10mM.

Description Chemical Properties Product Documents Related Products

MK-0249 is a potent histamine H3 receptor antagonist, with Ki of 1.7 nM for human H3.

[1]. Brioni JD, et al. Discovery of histamine H3 antagonists for the treatment of cognitive disorders and Alzheimer's disease. J Pharmacol Exp Ther. 2011 Jan;336(1):38-46.

리뷰

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Average Rating: 5 ★★★★★ (Based on Reviews and 17 reference(s) in Google Scholar.)

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