Raloxifene 4'-Glucuronide (Synonyms: Ral-4’-Gluc) |
| Catalog No.GC44804 |
Le 4'-glucuronide de raloxifène est un métabolite principal du raloxifène.
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Cas No.: 182507-22-8
Sample solution is provided at 25 µL, 10mM.
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Raloxifene 4'-glucuronide is a metabolite of the selective estrogen receptor modulator raloxifene . It is formed from raloxifene via the UDP-glucuronosyltransferase (UGT) isoforms UGT1A1, UGT1A8, and UGT1A10. It binds to the estrogen receptor with an IC50 value of 370 nM. Raloxifene 4'-glucuronide inhibits the voltage-gated potassium channel Kv4.3 by 6.2 and 20.1% when used at concentrations of 10 and 30 µM, respectively.
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