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α1 adrenoceptor-MO-1

カタログ番号GC31237

α1 アドレナリン受容体-MO-1、S エナンチオマーは、アルファ 1 アドレナリン受容体に親和性があり、アルファ分解活性を示し、鎮痛作用を持っています。 R エナンチオマーよりも活性が高い。

Products are for research use only. Not for human use. We do not sell to patients.

α1 adrenoceptor-MO-1 化学構造

Cas No.: 161905-64-2

サイズ 価格 在庫数 個数
1mg
$937.00
在庫あり
5mg
$1,866.00
在庫あり
10mg
$3,171.00
在庫あり
20mg
$5,598.00
在庫あり

Tel:(909) 407-4943 Email: sales@glpbio.com

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Sample solution is provided at 25 µL, 10mM.

Product Documents

Quality Control & SDS

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Background

α1 adrenoceptor-MO-1, an S enantiomer, has affinity at alpha 1 adrenergic receptor, shows alphalytic activity, and possesses analgesic action; more active than R enantiomer.

α1 adrenoceptor-MO-1 (the S enantiomer) and R enantiomer are more active than the corresponding racemates, but α1 adrenoceptor-MO-1 is more active than R enantiomer[1].

[1]. Pharmacologically active enantiomers. WO 1995001354 A1

Chemical Properties

Cas No. 161905-64-2 SDF
Canonical SMILES O=C1N(CCCN2[C@@H](C)CN(C3=CC=CC(Cl)=C3)CC2)N=C4C=CC=CN41
Formula C20H24ClN5O M.Wt 385.89
溶解度 Soluble in DMSO Storage Store at -20°C
General tips Please select the appropriate solvent to prepare the stock solution according to the solubility of the product in different solvents; once the solution is prepared, please store it in separate packages to avoid product failure caused by repeated freezing and thawing.Storage method and period of the stock solution: When stored at -80°C, please use it within 6 months; when stored at -20°C, please use it within 1 month.
To increase solubility, heat the tube to 37°C and then oscillate in an ultrasonic bath for some time.
Shipping Condition Evaluation sample solution: shipped with blue ice. All other sizes available: with RT, or with Blue Ice upon request.

Complete Stock Solution Preparation Table

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1 mg 5 mg 10 mg
1 mM 2.5914 mL 12.9571 mL 25.9141 mL
5 mM 0.5183 mL 2.5914 mL 5.1828 mL
10 mM 0.2591 mL 1.2957 mL 2.5914 mL
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計算

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO ( Master liquid concentration mg/mL, Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug. )

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Method for preparing in vivo formulation: Take μL DMSO master liquid, next add μL Corn oil, mix and clarify.

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Review for α1 adrenoceptor-MO-1

Average Rating: 5 ★★★★★ (Based on Reviews and 36 reference(s) in Google Scholar.)

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