Elacestrant S enantiomer dihydrochloride (Synonyms: RAD1901 S enantiomer dihydrochloride) |
カタログ番号GC60801 |
Elacestrant S 鏡像異性体二塩酸塩 (RAD1901 S 鏡像異性体二塩酸塩) は、Elacestrant 二塩酸塩の低活性鏡像異性体です。 Elacestrant (RAD1901) 二塩酸塩は、ERα および ERβ の IC50 値がそれぞれ 48 および 870 nM である、選択的かつ経口的に利用可能なエストロゲン受容体 (ERR) 分解剤です。
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Cas No.: 2309762-30-7
Sample solution is provided at 25 µL, 10mM.
Elacestrant S enantiomer dihydrochloride (RAD1901 S enantiomer dihydrochloride) is an low activity enantiomer of elacestrant dihydrochloride. Elacestrant (RAD1901) dihydrochloride is a selective and orally available estrogen receptor (ERR) degrader with IC50 values of 48 and 870 nM for ERα and ERβ, respectively.
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