M-144 |
| カタログ番号GC44107 |
UR-144は、末梢カンナビノイド（CB2）受容体（Ki = 1.8 nM）に中枢カンナビノイド（CB1）受容体（Ki = 150 nM）よりも選択的に結合する強力な合成カンナビノイドです。
Products are for research use only. Not for human use. We do not sell to patients.
Sample solution is provided at 25 µL, 10mM.
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UR-144 is a potent synthetic cannabinoid (CB) which preferentially binds the peripheral cannabinoid (CB2) receptor (Ki = 1.8 nM) over the central cannabinoid (CB1) receptor (Ki = 150 nM). [1] M-144 differs from UR-144 by having a fluorine atom on the terminal carbon of the alkyl group as well as a methyl group attached to the C2 carbon of the indole. The biological activities of this compound have not been characterized. This product is intended for forensic and research applications.
Reference:
[1]. Frost, J.M., Dart, M.J., Tietje, K.R., et al. Indol-3-ylcycloalkyl ketones: Effects of N1 substituted indole side chain variations on CB2 cannabinoid receptor activity. J. Med. Chem. 53(1), 295-315 (2010).
Average Rating: 5 (Based on Reviews and 36 reference(s) in Google Scholar.)
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