(Pen⁵)-Urotensin II (4-11) (human) |
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カタログ番号GA20269
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ペン-ウロテンシンII(4-11)(ヒト)(P5U)は、これまで報告された中で最も強力なウロテンシンII受容体アゴニストです。競争実験で測定された受容体に対する親和性は、ヒトのウロテンシンII(H-4768)より3倍高いことが示されています。P5Uは、人間のウロテンシンII/オーファング蛋白質共役受容体GPR14系の研究に有用なツールを提供する可能性があります。
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 473902-31-7
Sample solution is provided at 25 µL, 10mM.
(Pen5)-Urotensin II (4-11) (human) (P5U) is the most potent urotensin-II receptor agonist reported to date. It has been shown to exhibit a 3-fold higher affinity for the receptor (measured in competition experiments) than urotensin-II (human). P5U migh
| Cas No. | 473902-31-7 | SDF | |
| Formula | C52H68N10O12S2 | M.Wt | 1089.3 |
| 溶解度 | Soluble in DMSO | Storage | Store at -20°C |
| General tips | Please select the appropriate solvent to prepare the stock solution according to the
solubility of the product in different solvents; once the solution is prepared, please store it in
separate packages to avoid product failure caused by repeated freezing and thawing.Storage method
and period of the stock solution: When stored at -80°C, please use it within 6 months; when stored
at -20°C, please use it within 1 month. To increase solubility, heat the tube to 37°C and then oscillate in an ultrasonic bath for some time. |
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| Shipping Condition | Evaluation sample solution: shipped with blue ice. All other sizes available: with RT, or with Blue Ice upon request. | ||
| Prepare stock solution | |||
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1 mg | 5 mg | 10 mg |
| 1 mM | 918 μL | 4.5901 mL | 9.1802 mL |
| 5 mM | 183.6 μL | 918 μL | 1.836 mL |
| 10 mM | 91.8 μL | 459 μL | 918 μL |
Step 1: Enter information below (Recommended: An additional animal making an allowance for loss during the experiment)
Step 2: Enter the in vivo formulation (This is only the calculator, not formulation. Please contact us first if there is no in vivo formulation at the solubility Section.)
Calculation results:
Working concentration: mg/ml;
Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO ( Master liquid concentration mg/mL, Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug. )
Method for preparing in vivo formulation: Take μL DMSO master liquid, next addμL PEG300, mix and clarify, next addμL Tween 80, mix and clarify, next add μL saline, mix and clarify.
Method for preparing in vivo formulation: Take μL DMSO master liquid, next add μL Corn oil, mix and clarify.
Note: 1. Please make sure the liquid is clear before adding the next solvent.
2. Be sure to add the solvent(s) in order. You must ensure that the solution obtained, in the previous addition, is a clear solution before proceeding to add the next solvent. Physical methods such as vortex, ultrasound or hot water bath can be used to aid dissolving.
3. All of the above co-solvents are available for purchase on the GlpBio website.
Quality Control & SDS
- View current batch:
- Purity: >98.00% Appearance: A solid
- COA (Certificate of Analysis)
- SDS (Safety Data Sheet)
- Datasheet
Average Rating: 5 (Based on Reviews and 23 reference(s) in Google Scholar.)















