Perlapine (Synonyms: 6-(4-Methyl-1-piperazinyl)morphanthridine, NSC 291840) |
| カタログ番号GC44601 |
ペルラピンは強力なムスカリン性 DREADD (Designer Receptors Exclusively Activated by Designer Drugs) アゴニストであり、hM3 受容体よりも hM3Dq に対して >10000 倍の選択性を示します 。
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Cas No.: 1977/11/3
Sample solution is provided at 25 µL, 10mM.
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Perlapine is an atypical neuroleptic that blocks dopamine and serotonin (5-HT) receptors (Kis = 60, 30, and 30 nM for D2, D4, and 5-HT2A, respectively). Perlapine is also an agonist for hM3Dq, a designer receptor exclusively activated by designer drugs (DREADDs) derived from the human muscarinic acetylcholine M3 receptor that activates neuronal firing. Perlapine displays >10,000-fold selectivity for hM3Dq over hM3.
Average Rating: 5 (Based on Reviews and 33 reference(s) in Google Scholar.)
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