H-Tyr-Cys-Phe-Ala-Trp-Lys-Thr-Phe-Cys-OH |
Catalog No.GA22966 |
Selective somatostatin receptor subtype sst4 agonist. In competitive radioligand displacement experiments using the non-selective radioligand ([¹²?I]-(Leu?,D-Trp²²,Tyr²?)-Somatostatin-28, YCFAWKTFC exhibited a high affinity for sst4 with an IC?? value of 2.0 ± 0.5 nM. IC?? values for sst1, sst2, sst3, and sst5 were >1000 nM, 622 ± 85 nM, 624 ± 213 nM, and 692 ± 166 nM, respectively. The nonapeptide YCFAWKTFC may serve as a lead compound or tool for preclinical and clinical studies.
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Cas No.: 647016-22-6
Sample solution is provided at 25 µL, 10mM.
Selective somatostatin receptor subtype sst4 agonist. In competitive radioligand displacement experiments using the non-selective radioligand ([¹²I]-(Leu,D-Trp²²,Tyr²)-Somatostatin-28, YCFAWKTFC exhibited a high affinity for ss
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