Other Signal Transduction
Signal Transduction
Cellular responses are triggered by proteins, drugs, or pathogens binding to specific receptors. Receptor mediated signaling is a cascade of enzymatic reactions that amplifies the signal. The agonists and antagonists modulating receptor functionality are essential tools for research and medical practice. read more
Targets for Other Signal Transduction
Products for Other Signal Transduction
- Cat.No. 상품명 정보
-
GC49890
β-Glycerophosphate-d5 (sodium salt hydrate)
Glycerol 2-Phosphate-d5
An internal standard for the quantification of β-glycerophosphate -
GC13863
10Panx
10Panx
A peptide inhibitor of PANX1 -
GC49912
13C20,15N10-Cyclic di-GMP (sodium salt)
13C20,15N10-c-di-GMP, 13C20,15N10-Cyclic diguanylate, 13C20,15N10-3’,5’-Cyclic diguanylic Acid
An internal standard for the quantification of cyclic di-GMP - GC52141 2-Chloro-N-methyl-N-(4-nitrophenyl)acetamide
-
GC52129
3-Amino-5-hydroxybenzoic Acid
AHBA
-
GC49494
4-Aminobenzylphosphonic Acid
4-ABPA, NSC 12117
An alkaline phosphatase inhibitor -
GP10121
Ac-Endothelin-1 (16-21), human
Ac-His-Leu-Asp-Ile-Ile-Trp-OH
-
GP10059
Acetyl Angiotensinogen (1-14), porcine
Ac-Asp-Arg-Val-Tyr-Ile-His-Pro-Phe-His-Leu-Leu-Val-Tyr-Ser-OH
-
GP10076
Agouti-related Protein (AGRP) (25-82), human
H2N-Leu-Ala-Pro-Met-Glu-Gly-Ile-Arg-Arg-Pro-Asp-Gln-Ala-Leu-Leu-Pro-Glu-Leu-Pro-Gly-Leu-Gly-Leu-Arg-Ala-Pro-Leu-Lys-Lys-Thr-Thr-Ala-Glu-Gln-Ala-Glu-Glu-Asp-Leu-Leu-Gln-Glu-Ala-Gln-Ala-Leu-Ala-Glu-Val-Leu-Asp-Leu-Gln-Asp-Arg-Glu-Pro-Arg-OH
-
GC49110
AICA Ribonucleotide
AICA-Ribotide, AICA-Riboside-5'-phosphate, 5-Aminoimidazole-4-Carboxamide Ribonucelotide, NSC 283955, NSC 292227
An AMPK activator -
GC52361
AMARA Peptide (trifluoroacetate salt)
AMARAASAAALARRR-OH, H-Ala-Met-Ala-Arg-Ala-Ala-Ser-Ala-Ala-Ala-Leu-Ala-Arg-Arg-Arg-OH
A peptide substrate for AMPK -
GP10077
Angiotensin (1-7)
Asp-Arg-Val-Tyr-Ile-His-Pro
Ang-(1-7) (H - Asp - Arg - Val - Tyr - Ile - His - Pro - OH)는 내인성 펩타이드 단편으로, Ang I 또는 Ang II를 각각 endo- 또는 carboxy-peptidase를 통해 생산할 수 있습니다[1].
-
GP10074
Angiotensin 1/2 (1-5)
H2N-Asp-Arg-Val-Tyr-Ile-OH
-
GP10067
Angiotensin 1/2 (1-6)
H2N-Asp-Arg-Val-Tyr-Ile-His-OH
-
GP10144
Angiotensin 1/2 (1-7) amide
H2N-Asp-Arg-Val-Tyr-Ile-His-Pro-amide
-
GP10012
Angiotensin 1/2 (1-8) amide
H2N-Asp-Arg-Val-Tyr-Ile-His-Pro-Phe-amide
Vasoconstrictor
- GP10025 Angiotensin 1/2 (1-9)
-
GP10045
Angiotensin 1/2 (2-7)
H2N-Arg-Val-Tyr-Ile-His-Pro-OH
Vasoconstrictor
-
GP10079
Angiotensin 1/2 (5-7)
H2N-Ile-His-Pro-OH
-
GP10120
Angiotensin 1/2 + A (2 - 8)
H2N-Ala-Arg-Val-Tyr-Ile-His-Pro-Phe-OH
Vasoconstrictor - GP10087 Angiotensin I (human, mouse, rat)
-
GP10023
Angiotensin II
AT1 및 AT2 수용체에서의 작용제
- GP10110 Angiotensin III (human, mouse) An agonist at AT1 and AT2 receptors
-
GP10137
ANP (1-11), rat
H2N-Ser-Leu-Arg-Arg-Ser-Ser-Cys-Phe-Gly-Gly-Arg-OH
-
GP10061
Atrial Natriuretic Factor (1-29), chicken
H2N-Met-Met-Arg-Asp-Ser-Gly-Cys-Phe-Gly-Arg-Arg-Ile-Asp-Arg-Ile-Gly-Ser-Leu-Ser-Gly-Met-Gly-Cys-Asn-Gly-Ser-Arg-Lys-Asn-OH
Atrial Natriuretic Factor (1-29), chicken, (C130H223N51O41S5), a peptide with the sequence H2N-SPKMVQGSGCFGRKMDRISSSSGLGCKVLRRH-OH, MW= 3316.8. -
GC49403
Benzarone
L 2197, NSC 82134
Benzarone(Fragivix)은 난모세포에서 IC50이 2.8μM인 강력한 인간 요산 수송체 1(hURAT1) 억제제입니다. - GC49300 BIM-46187 (hydrochloride) An inhibitor of heterotrimeric G-protein signaling
-
GC19508
BLU-782
Activin Receptor-like Kinase 2 Inhibitor 1, ALK2-IN-1, Fidrisertib
BLU-782는 ALK2돌연변이를 치료하기 위해 경구 복용을 하는 정밀 치료법이다. - GP10071 BNP (1-32), human
- GC49079 C82 An Mtb CdnP inhibitor
-
GC49332
Calcineurin Substrate (trifluoroacetate salt)
H-Asp-Leu-Asp-Val-Pro-Ile-Pro-Gly-Arg-Phe-Asp-Arg-Arg-Val-Ser-Val-Ala-Ala-Glu-OH, H-DLDVPIPGRFDRRVSVAAE-OH
A synthetic peptide substrate - GC49433 Capsiate Capsiate는 매운맛이 없는 CH-19 sweet red pepper 품종에서 추출한 capsaicin 유사체로서 TRPV1의 경구 활성 작용제입니다.
- GC48992 CGP 77675 (hydrate) An inhibitor of Src family kinases
-
GC49392
CHIR98024
CT 98024
CHIR98024(화합물 L)는 0.2566μM의 EC50을 갖는 글리코겐 합성효소 키나제 3(GSK3) 억제제입니다. -
GC49334
Chroman 1 (hydrochloride hydrate)
(S)-Chroman 1
A ROCK2 inhibitor -
GC49556
Cl-Necrostatin-1
7-Cl-Nec-1, 7-Cl-Necrostatin-1, Nec-1f
A RIPK1 inhibitor -
GP10134
coagulation factor II (thrombin) B chain fragment [Homo sapiens]
H2N-Lys-Pro-Val-Ala-Phe-Ser-Asp-Tyr-Ile-His-Pro-Val-Cys-Leu-Pro-Asp-Arg-OH
-
GP10010
COG 133
Leu-Arg-Val-Arg-Leu-Ala-Ser-His-Leu-Arg-Lys-Leu-Arg-Lys-Arg-Leu-Leu
-
GC49789
Dihydronarwedine
(–)-Dihydrogalanthaminone, (–)-Lycoraminone
An alkaloid and GSK3β inhibitor -
GP10022
Dynamin inhibitory peptide
Gln-Val-Pro-Ser-Arg-Pro-Asn-Arg-Ala-Pro
-
GC13855
Eeyarestatin I
엔도플라즘질망 연관 분해(ERAD) 및 단백질 이동의 억제제
-
GP10030
EGF receptor substrate eps15 acetyl - [Mus musculus]/[Homo sapiens]
Ac-Gln-Glu-Gln-Glu-Asp-Leu-Glu-Leu-Ala-Ile-Ala-Leu-Ser-Lys-Ser-Glu-Ile-Ser-Glu-Ala-OH
EGF receptor substrate eps15 (Eps15) has been identified as a 142-kDa substrate of the EGF receptor1. -
GP10108
EGF-R (661-681) T669 Peptide
H2N-Lys-Arg-Glu-Leu-Val-Glu-Pro-Leu-Thr-Pro-Ser-Gly-Glu-Ala-Pro-Asn-Gln-Ala-Leu-Leu-Arg-OH
-
GC52002
Emavusertib
CA-4948
Emavusertib(CA-4948)은 항종양 활성이 있는 강력한 IRAK4/FLT3 억제제입니다. - GP10065 Endomorphin-1
-
GP10117
Endostatin (84-114)-NH2 (JKC367)
H2N-Pro-Gly-Ala-Arg-Ile-Phe-Ser-Phe-Asp-Gly-Lys-Asp-Val-Leu-Arg-His-Pro-Thr-Trp-Pro-Gln-Lys-Ser-Val-Trp-His-Gly-Ser-Asp-Pro-Asn-NH2
-
GP10062
Endothelin-1 (1-15), amide, human
H2N-Cys-Ser-Cys-Ser-Ser-Leu-Met-Asp-Lys-Glu-Cys-Val-Tyr-Phe-Cys-NH2
- GC52336 ENPP1 Inhibitor 43 An ENPP1 inhibitor
- GC52277 ENPP3 Inhibitor An ENPP3 inhibitor
- GC52362 ENPP3 Inhibitor 4g An ENPP1 and ENPP3 inhibitor
- GC52322 ENPP3 Inhibitor 4t An ENPP3 inhibitor
-
GP10005
Epidermal growth factor receptor (994-1002) acetyl/amide
Ac-Asp-Ser-Asn-Phe-Tyr-Arg-Ala-Leu-Met-amide
EGF-family receptor
-
GP10095
Epidermal Growth Factor Receptor Peptide (985-996)
H2N-Asp-Val-Val-Asp-Ala-Asp-Glu-Tyr-Leu-Ile-Pro-Gln-OH
-
GP10132
erbB-2
H2N-Lys-Ile-Phe-Gly-Ser-Leu-Ala-Phe-Leu-OH
- GC49074 Forphenicine A bacterial metabolite and an inhibitor of alkaline phosphatase
-
GP10092
G protein coupled receptor [Homo sapiens]
H2N-Gln-Glu-Ser-His-Asn-Ser-Gly-Asn-Arg-Ser-Asp-Gly-Pro-Gly-Lys-Asn-Thr-Thr-Leu-His-Asn-Glu-Phe-Asp-Thr-OH
G protein coupled receptor [Homo sapiens], (C110H168N38O45), a peptide with the sequence H2N-QESHNSGNRSDGPGKNTTLHNEFDT-OH, MW= 2742.74. -
GP10107
Gap 26
Val-Cys-Tyr-Asp-Lys-Ser-Phe-Pro-Ile-Ser-His-Val-Arg
-
GP10119
Gap 27
Ser-Arg-Pro-Thr-Glu-Lys-Thr-Ile-Phe-Ile-Ile
A connexin-mimetic peptide
-
GC25450
GATA4-NKX2-5-IN-1
3i-1000
GATA4-NKX2-5-IN-1 (3i-1000) is a small-molecule compound inhibiting GATA4 and NKX2-5 transcriptional synergy with IC50 of 3 uM
-
GP10122
Glucagon (19-29), human
H2N-Ala-Gln-Asp-Phe-Val-Gln-Trp-Leu-Met-Asn-Thr-OH
-
GP10024
Growth Hormone (1-43), human
H2N-Phe-Pro-Thr-Ile-Pro-Leu-Ser-Arg-Leu-Phe-Asp-Asn-Ala-Met-Leu-Arg-Ala-His-Arg-Leu-His-Gln-Leu-Ala-Phe-Asp-Thr-Tyr-Gln-Glu-Phe-Glu-Glu-Ala-Tyr-Ile-Pro-Lys-Glu-Gln-Lys-Tyr-Ser-OH
Human Growth Hormone (1-43) peptide - GC49284 GSK-A1 GSK-A1은 pIC50이 8.5-9.8인 선택적 III형 포스파티딜이노시톨 4-키나제 PI4KA(PI4KIIIα) 억제제입니다.
-
GP10004
GTP binding protein 1 fragment [Multiple species]
H2N-Lys-Val-Ile-Thr-Phe-Ile-Asp-Leu-OH
Signal transducing molecules -
GP10115
GTP-Binding Protein Fragment, G alpha
H2N-Cys-Gly-Ala-Gly-Glu-Ser-Gly-Lys-Ser-Thr-Ile-Val-Lys-Gln-Met-Lys-OH
-
GP10041
Insulin like growth factor II fragment variant
H2N-Thr-Pro-Thr-Lys-Ser-Glu-Arg-OH
Insulin like growth factor II fragment variant has a sequence of Thr-Pro-Thr-Lys-Ser-Glu-Arg. -
GP10029
Interleukin II (60-70)
H2N-Leu-Thr-Phe-Lys-Phe-Tyr-Met-Pro-Lys-Lys-Ala-OH
Cytokine,regulating WBC
-
GC52328
KYL (trifluoroacetate salt)
KYL Peptide
An EphA4 inhibitor -
GC17779
Levetiracetam
UCBL 059
항간질제인 레베티라세탐은 시냅스 소포 단백질 SV2A에 결합합니다. -
GP10140
MAP kinase fragment [Multiple species]
H2N-Lys-Tyr-Ile-His-Ser-Ala-Asn-Val-Leu-OH
-
GP10066
Melanocyte stimulating hormone release inhibiting factor
Pro-Leu-Gly
-
GC49269
Myr-ZIP
Myristoylated-ZIP, Myristoylated Zeta-Pseudosubstrate Inhibitory Peptide, Myr-Ser-Ile-Tyr-Arg-Arg-Gly-Ala-Arg-Arg-Trp-Arg-Lys-Leu, Myr-SIYRRGARRWRKL-OH, Ζeta Inhibitory Peptide
A PKMζ inhibitor -
GC49090
Nilvadipine-d4
(±)-Nilvadipine-d4
An internal standard for the quantification of nilvadipine -
GP10011
Nitric Oxide Synthase (599-613) Blocking Peptide, Bovine Endothelial Cell
Ac-Pro-Tyr-Asn-Ser-Ser-Pro-Arg-Pro-Glu-Gln-His-Lys-Ser-Tyr-Lys-Cys-OH
- GP10069 Parathyroid hormone (1-34) (human)
-
GC52151
PKCθ Inhibitor (hydrochloride)
Protein Kinase C θ Inhibitor
-
GC49265
PKI (14-22) amide (myristoylated) (trifluoroacetate salt)
Myr-Gly-Arg-Thr-Gly-Arg-Arg-Asn-Ala-Ile-NH2, Myr-GRTGRRNAI-NH2, Myristoylated PKI-(14-22)-amide, PKI-(Myr-14-22)-amide
A PKA inhibitor -
GP10053
Prothrombin (474-477) [Mus musculus]
H2N-Tyr-Ile-His-Pro-OH
- GC49221 QLT0267 An ILK inhibitor
-
GP10042
Rhodopsin peptide
H2N-Val-Ser-Lys-Thr-Glu-Thr-Ser-Gln-Val-Ala-Pro-Ala-OH
- GC52115 S-99 An inhibitor of ASK1
-
GP10104
S6 Kinase Substrate Peptide 32
H2N-Lys-Glu-Ala-Lys-Glu-Lys-Arg-Gln-Glu-Gln-Ile-Ala-Lys-Arg-Arg-Arg-Leu-Ser-Ser-Leu-Arg-Ala-Ser-Thr-Ser-Lys-Ser-Gly-Gly-Ser-Gln-Lys-OH
Measures the activity of kinases that phosphorylate ribosomal protein S6. -
GC11058
Scrambled 10Panx
Scrambled 10Panx Phe-Ser-Val-Tyr-Trp-Ala-Gln-Ala-Asp-Arg
Panx-1 mimetic inhibitory peptide, blocks pannexin-1 gap junctions
-
GP10093
signal transducer and activator of transcription 5 (322-343) acetyl/amide
Ac-Asp-Ile-Ile-Ser-Ala-Leu-Val-Thr-Ser-Thr-Phe-Ile-Ile-Glu-Lys-Gln-Pro-Pro-Gln-Val-Leu-Lys-amide
signal transducer and activator of transcription 5 (322-343) acetylamide, (C115H193N27O33), a peptide with the sequence Ac-DIISALVTSTFIIEKQPPQVLK-amide, MW= 2481.92. -
GP10145
signal transducer and activator of transcription 6 fragment
H2N-Ser-Tyr-Trp-Ser-Asp-Arg-Leu-Ile-Ile-OH
-
GP10085
Thrombin Receptor Activator for Peptide 5 (TRAP-5)
H2N-Ser-Phe-Leu-Leu-Arg-OH
-
GC49692
Tofacitinib-d3 (citrate)
CP 690,550-d3
An internal standard for the quantification of tofacitinib -
GC49150
Tpl2 Kinase Inhibitor (hydrochloride)
c-Cot Kinase Inhibitor, MAP3K8 Kinase Inhibitor, Tumor Progression Locus 2 Kinase Inhibitor
A Tpl2 inhibitor -
GP10112
TRH Precursor Peptide
H2N-Lys-Arg-Gln-His-Pro-Gly-Lys-Arg-OH
Thyrotropin Releasing Hormone Precursor Peptide
-
GP10091
Vasonatrin Peptide (1-27)
H2N-Gly-Leu-Ser-Lys-Gly-Cys-Phe-Gly-Leu-Lys-Leu-Asp-Arg-Ile-Gly-Ser-Met-Ser-Gly-Leu-Gly-Cys-Asn-Ser-Phe-Arg-Tyr-OH
Vasonatrin Peptide (1-27), (C124H198N36O36S3), a peptide with the sequence H2N-GLSKGCFGLKLDRIGSMSGLGCNSFRY-OH, MW= 2865.4. -
GC52274
Y-33075 (hydrochloride)
RKI-983, SNJ-1656, Y-39983
An inhibitor of ROCK2 -
GP10017
[Ser25] Protein Kinase C (19-31)
H2N-Arg-Phe-Ala-Arg-Lys-Gly-Ser-Leu-Arg-Gln-Lys-Asn-Val-OH
PKC substrate
-
GP10096
β-Interleukin I (163-171), human
H2N-Val-Gln-Gly-Glu-Glu-Ser-Asn-Asp-Lys-OH
-
GP10080
β-Interleukin II (44-56)
H2N-Ile-Leu-Asn-Gly-Ile-Asn-Asn-Tyr-Lys-Asn-Pro-Lys-Leu-OH
-
GP10111
β-Pompilidotoxin
Arg-Ile-Lys-Ile-Gly-Leu-Phe-Asp-Gln-Leu-Ser-Arg-Leu