Target Protein-binding moiety 4 (Synonyms: Molibresib carboxylic acid; GSK525762A carboxylic acid; PROTAC BRD4-binding moiety 2) |
| Catalog No.GC32863 |
El resto de uniÓn a proteÍnas diana 4 (Ácido carboxÍlico de molibresib) es un ligando de ojiva basado en I-BET762 para reacciones de conjugaciÓn de PROTAC dirigido a BET. El resto de uniÓn a proteÍnas diana 4 (Ácido carboxÍlico de molibresib) es un inhibidor de BRD4 con una pIC50 de 5,1.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 1300019-38-8
Sample solution is provided at 25 µL, 10mM.
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Target Protein-binding moiety 4 is a BRD4(1) inhibitor with an IC50 of 7.9 μM.
Target Protein-binding moiety 4 (compound 32) is a BRD4 (1) inhibitor with an IC50 of 7.9 μM[1].
[1]. Yifei Yang, et al. Combined pharmacophore models as virtual screening protocol against BRD4(1) inhibitor. Medicinal Chemistry Research (2016), 25(4), 585-595.
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