Target Protein-binding moiety 4 (Synonyms: Molibresib carboxylic acid; GSK525762A carboxylic acid; PROTAC BRD4-binding moiety 2) |
| Katalog-Nr.GC32863 |
Die Zielprotein-bindende Einheit 4 (Molibresib-CarbonsÄure) ist ein I-BET762-basierter Gefechtskopf-Ligand fÜr Konjugationsreaktionen von PROTAC-Targeting auf BET. Zielprotein-bindende Einheit 4 (Molibresib-CarbonsÄure) ist ein BRD4-Inhibitor mit einem pIC50 von 5,1.
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Cas No.: 1300019-38-8
Sample solution is provided at 25 µL, 10mM.
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Target Protein-binding moiety 4 is a BRD4(1) inhibitor with an IC50 of 7.9 μM.
Target Protein-binding moiety 4 (compound 32) is a BRD4 (1) inhibitor with an IC50 of 7.9 μM[1].
[1]. Yifei Yang, et al. Combined pharmacophore models as virtual screening protocol against BRD4(1) inhibitor. Medicinal Chemistry Research (2016), 25(4), 585-595.
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