GLPBio

GPCR/G protein

Research Areas

Products Related to GPCR/G protein(3538)

  • GC74416 structure
    GC74416P4pal10 TFA
    Purity: >98.00%

    P4pal10 TFA هو شكل ملح TFA من P4pal10.

  • GC74478 structure
    GC74478Ulocuplumab
    CAS: 1375830-34-4
    Purity: >99.00%

    Ulocuplumab (مضاد للبشر CXCR4 المؤتلف/BMS-936564/MDX1338) هو جسم مضاد لـ CXCR4 كامل الجسم البشري.

  • GC74632 structure
    GC74632Benzquinamide hydrochloride
    CAS: 113-69-9
    Purity: >99.00%

    Benzquinamide hydrochloride (P2647) هو مضاد للقيء الذي يمكن أن يرتبط مع مستقبلات α2A و α2B و α2C الأدرينالية (α2-AR) مع قيم Ki من 1,365 و 691 و 545 نانومتر، على التوالي.

  • GC74636 structure
    GC74636GR 55562 hydrochloride
    CAS: 172854-55-6
    Purity: >98.00%

    GR 55562 hydrochloride هو انتقائية 5-HT1B مضاد مستقبلات.

  • GC74667 structure
    GC74667GPR109 receptor agonist-2
    CAS: 957129-38-3
    Purity: >99.00%

    GPR109 receptor agonist-2 (المركب 5) هو ناشر انتقائي GPR109a مع pEC50 من 5.53.

  • GC78786 structure
    GC78786Z52-L16
    CAS: 3077488-80-0
    Purity: >98.00%

    Z52 -L16 is Drug-Linker Conjugates for ADC, which is composed of a linker and a Ras inhibitor Z52.

  • GC78913 structure
    GC78913Antiparasitic agent-30
    CAS: 671754-20-4
    Purity: >98.00%

    Antiparasitic agent-30 is a potent adenosine kinase TbrAK modulator and antitrypanosomal agent.

  • GC79165 structure
    GC79165Snail IN-1
    CAS: 3083216-69-4
    Purity: >98.00%

    Snail IN-1 is an orally active Snail inhibitor with a Ka of 0.36 μM.Snail IN-1 disrupts Snail - CBP interaction, accelerates Snail protein degradation, reduces Snail acetylation, increases Snail polyubiquitination, and selectively downregulates Snail protein without altering other EMT transcription factors.Snail IN-1 reduces atherosclerotic plaque burden, modulates inflammation and plaque stability factors, downregulates CCL5, CXCL10, MMP2, and MMP9, and upregulates α-smooth muscle actin.Snail IN-1 exerts anti-inflammatory and plaque-stabilizing properties.Snail IN-1 can be used for the research of atherosclerosis [1] .

  • GC79166 structure
    GC79166Zilebesiran
    CAS: 2380166-33-4
    Purity: >95.50%

    Zilebesiran is a siRNA that reduce hepatic angiotensinogen levels through RNA interference.

  • GC79190 structure
    GC79190IRFI-165
    CAS: 191349-26-5
    Purity: >98.00%

    IRFI-165 is a potent and selective A 1 adenosine receptor antagonist with a K i of 7.9 nM for rat A 1 AR.

  • GC79191 structure
    GC79191EXP-7711
    CAS: 114798-27-5
    Purity: >99.00%

    EXP-7711 is a non peptide angiotensin II (Ang II) AT1 receptor antagonist.

  • GC79192 structure
    GC79192L-161638
    CAS: 150484-73-4
    Purity: >98.00%

    L-161638 is a potent, selective and orally active AT2 receptor antagonist.

  • GC79193 structure
    GC79193(Des-Asp1,Ile8)-Angiotensin II
    CAS: 52498-25-6
    Purity: >98.50%

    (Des-Asp1,Ile8)-Angiotensin II is a peptide related to angiotensin II.

  • GC79194 structure
    GC79194Exendin-4-Cys
    Purity: >99.50%

    Exendin-4 -Cys is a cysteine-modified Exendin-4.

  • GC79195 structure
    GC79195Semaglutide-FITC
    Purity: >96.50%

    Semaglutide -FITC (Semaglutide-Lys(FITC)) is a fluorescent tracer probe (Ex/Em = 495/520 nm) obtained by covalently coupling the green fluorescent dye fluorescein isothiocyanate (FITC) to the long-acting analogue of GLP-1, Semaglutide.

  • GC79196 structure
    GC79196Semaglutide, Cy5 labeled
    Purity: >98%

    Semaglutide, Cy5-labeled (Semaglutide-Cys(Cy5)) is a CY5 -labeled version of Semaglutide (Ex/Em = 633/670 nm).

  • GC79197 structure
    GC79197Gamma-Glu-Abu acetate
    Purity: >99.50%

    Gamma-Glu-Abu acetate is a CaSR activator with an EC 50 of 0.21 μM (in HEK-293 cells).

  • GC79198 structure
    GC79198KP-2067
    CAS: 1262781-19-0
    Purity: >98%

    KP-2067 is a form of the CaSR agonist peptide.

  • GC79199 structure
    GC79199[Tyr0] Corticotropin Releasing Factor, ovine acetate
    Purity: >98.00%

    [Tyr0] Corticotropin Releasing Factor, ovine acetate is a corticotropin releasing factor/hormone isolated from ovine.

  • GC79200 structure
    GC79200Annexuzlimab
    Purity: >98.50%

    Annexuzlimab is a humanised IgG1 monoclonal antibody which specifically binds to ANXA1 disrupting its interaction with formyl peptide receptors 1 and 2 (FPR1/2).

  • GC79201 structure
    GC79201TUG-2304
    CAS: 3034674-48-8
    Purity: >98.50%

    TUG-2304 is a highly selective free fatty acid receptor 2 ( FFA2, GPR43 ) antagonist that completely suppresses propionate-induced neutrophil migration and respiratory burst.

  • GC79202 structure
    GC79202LY3324954
    Purity: >98.50%

    LY3324954 is a long-acting, highly selective glucagon receptor ( GCGR ) agonist.

  • GC79203 structure
    GC79203GIPR antagonist 1
    CAS: 3059497-30-9
    Purity: >98%

    GIPR antagonist 1 is a GIPR antagonist with an IC 50 of 4.8 nM.

  • GC79204 structure
    GC79204(S)-PF-5190457
    Purity: >99.00%

    (S)-PF-5190457 ((S)-PF-05190457) is the S-enantiomer of PF-5190457.