GPCR/G protein
Research Areas
- Neuropeptide FF/AF Receptors(51)
- Neuropeptide S Receptor(3)
- GPBA Receptor(3)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- Formyl Peptide Receptors(11)
- 5-HT Receptor(414)
- Acetylcholine(28)
- Adenosine Deaminase(10)
- Adenosine Receptor(138)
- Adenosine Kinase(5)
- Adiponectin Receptor(3)
- Adrenergic Receptor(431)
- Adrenergic Transporters(5)
- Apelin Receptor(9)
- Angiotensin Receptor(117)
- Bombesin Receptors(23)
- Bradykinin Receptors(29)
- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(111)
- Calcimimetic Agent(2)
- CaSR(25)
- CCK1 Receptors(7)
- CCK2 Receptors(7)
- CCR(95)
- Chemokine Receptors(23)
- CRF1 Receptors(10)
- CRF2 Receptors(3)
- CXCR(93)
- CysLT1 receptor(1)
- Endothelin Receptor(53)
- EP1 Receptor(2)
- EP4 Receptor(2)
- ERRγ(1)
- ETA Receptors(5)
- ETB Receptors(5)
- Free Fatty Acid Receptors(16)
- Galanin Receptors(11)
- Ghrelin Receptors(11)
- GHSR(20)
- GIP Receptor(5)
- Glucagon Receptor(54)
- Glucocorticoid Receptor(94)
- GLUT1(1)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(12)
- GPR109A(4)
- GPR119(10)
- GPR120(9)
- GPR35(10)
- GPR44(1)
- GPR55(11)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(57)
- LPA Receptor(12)
- LPL Receptor(62)
- LTD4 Receptor(1)
- mGluR (123)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(57)
- Melatonin Receptors(23)
- Motilin Receptor(7)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(26)
- NK2 Receptors(7)
- NK3 Receptor(5)
- NOP Receptor(20)
- NPY Receptors(26)
- Orexin(3)
- Orphan 7-TM Receptors(6)
- OX Receptor(52)
- Oxytocin Receptors(22)
- P2Y Receptor(65)
- PACAP Receptors(7)
- PAF Receptors(7)
- Peptide Receptors(14)
- PGD2 Receptor(1)
- Prostaglandin Receptor(174)
- Prostanoid Receptors(25)
- Protease-Activated Receptors(9)
- RGS(2)
- S1P receptor(8)
- Secretin Receptors(1)
- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(43)
- Sigma Receptor(59)
- Vasopressin Receptor(34)
- 17,20-lyase(4)
- Ras(163)
- Urotensin-II Receptor(10)
- VIP Receptors(6)
- EBI2/GPR183(7)
- TSH Receptor(10)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(20)
- GPR84(10)
- Neuromedin U Receptors(2)
- Kisspeptin Receptor(6)
- CRFR(27)
- RGS Protein(5)
- Urotensin Receptor(7)
- Cholecystokinin Receptor(28)
- GPR139(4)
- mAChR(191)
- MCHR1 (GPR24)(16)
- Neurokinin Receptor(76)
- cGMP(27)
- GRK(3)
- GPR88(1)
- Amylin Receptor(3)
- Arrestin(8)
- Mas-related G-protein-coupled Receptor (MRGPR)(6)
- GCGR(7)
- GLP Receptor(16)
- Succinate Receptor 1(1)
- PTHR(2)
- Protease Activated Receptor (PAR)(6)
- Free Fatty Acid Receptor(5)
- Formyl Peptide Receptor (FPR)(3)
- Hydroxycarboxylic Acid Receptor (HCAR)(2)
- RXFP Receptor(2)
- Adhesion G Protein-coupled Receptors (AGPCRs)(1)
- Taste Receptor(1)
- GPR52(1)
Products Related to GPCR/G protein(3538)
- GC81704Ractopamine-d 6CAS: 1185177-97-2Purity: >98%
Ractopamine -d 6 is the deuterium labeled Ractopamine.
- GC81729Neuropeptide W-30 (rat) acetatePurity: >98.00%
Neuropeptide W-30 (rat) is an important stress mediator in the central nervous system that modulates the hypothalamus-pituitary-adrenal (HPA) axis and sympathetic outflow.
- GC817573-Ethoxy-5,6-dibromosalicylaldehydeCAS: 20041-64-9Purity: >99.50%
3-Ethoxy-5,6-dibromosalicylaldehyde is an IRE1/ERN1 inhibitor, with an IC 50 of 0.12 μM, a K i of 71-88 nM, and a K d of 100 nM against the ribonuclease activity of hIRE1α, as well as an IC 50 of 4.8 μM against yeast Ire1.
- GC81851Pancreatic Polypeptide, rat TFAPurity: >98.00%
Pancreatic Polypeptide, rat TFA (Rat pancreatic polypeptide TFA) is a rat-derived Pancreatic Polypeptide.
- GC81855(R)-RXFP2 agonist 2CAS: 3123585-08-7Purity: >98.00%
(R)-RXFP2 agonist 2 is the R-type isomer of RXFP2 agonist 2.
- GC81859TH-Z827 diTFAPurity: >98.00%
TH-Z827 diTFA is a selective KRAS G12D inhibitor that exhibits activity against GDP-bound and GMPPNP-bound KRAS G12D, but shows no activity against KRAS (WT) and KRAS G12C.
- GC81870Bethanidine hydriodideCAS: 2863-34-5Purity: >98.00%
Bethanidine hydriodide is an orally active antihypertensive agent and adrenergic neuron blocker.
- GC909521-Aminoguanosine-3',5'-monophosphate (sodium salt)CAS: 1380911-23-8Purity: >95.00%
مادة أساسية لإنزيم بروتين كيناز الـ cGMP-المعتمد.
- GC92078PKG Inhibitor (trifluoroacetate salt)Purity: >95.00%
PKG Inhibitor (trifluoroacetate salt) هو مثبط يعتمد على cGMP PKG Ki = 86 ميكرومتر.
| Catalog No. | Product Name | CAS No. | Purity | Structure |
|---|---|---|---|---|
| GC81704 | Ractopamine-d 6 | 1185177-97-2 | >98% | |
Ractopamine -d 6 is the deuterium labeled Ractopamine. | ||||
| GC81727 | HOR1-C59 | 189574-20-7 | >99.50% | |
HOR1-C59 is a highly selective Or5v1/Olfr110 agonist with an EC 50 of 7.12 nM. | ||||
| GC81728 | TTFB | 352560-76-0 | >98.00% | |
TTFB (N-(4-tert-butyl-1,3-thiazol-2-yl)-3-fluorobenzamide) is a selective, non-competitive zinc-activated channel ( ZAC ) antagonist. | ||||
| GC81729 | Neuropeptide W-30 (rat) acetate | - | >98.00% | |
Neuropeptide W-30 (rat) is an important stress mediator in the central nervous system that modulates the hypothalamus-pituitary-adrenal (HPA) axis and sympathetic outflow. | ||||
| GC81739 | LY 78335 | 39226-94-3 | >99.00% | |
LY 78335 (DCMB) is a brain-penetrant phenylethanolamine-N-methyltransferase ( PNMT ) inhibitor with a K i of 0.09 μM. | ||||
| GC81757 | 3-Ethoxy-5,6-dibromosalicylaldehyde | 20041-64-9 | >99.50% | |
3-Ethoxy-5,6-dibromosalicylaldehyde is an IRE1/ERN1 inhibitor, with an IC 50 of 0.12 μM, a K i of 71-88 nM, and a K d of 100 nM against the ribonuclease activity of hIRE1α, as well as an IC 50 of 4.8 μM against yeast Ire1. | ||||
| GC81769 | LP-856866 | - | >99.50% | |
LP-856866 is an orally active ACSL5 inhibitor, with IC 50 values of 8 nM and 4 nM against mouse and human ACSL5, respectively, and IC 50 values of 6 nM and 17 nM against mouse and human ACSL1, respectively. | ||||
| GC81824 | (+)-Talinolol | 71369-60-3 | >99.00% | |
(+)-Talinolol is an isomer of Talinolol. | ||||
| GC81851 | Pancreatic Polypeptide, rat TFA | - | >98.00% | |
Pancreatic Polypeptide, rat TFA (Rat pancreatic polypeptide TFA) is a rat-derived Pancreatic Polypeptide. | ||||
| GC81855 | (R)-RXFP2 agonist 2 | 3123585-08-7 | >98.00% | |
(R)-RXFP2 agonist 2 is the R-type isomer of RXFP2 agonist 2. | ||||
| GC81859 | TH-Z827 diTFA | - | >98.00% | |
TH-Z827 diTFA is a selective KRAS G12D inhibitor that exhibits activity against GDP-bound and GMPPNP-bound KRAS G12D, but shows no activity against KRAS (WT) and KRAS G12C. | ||||
| GC81870 | Bethanidine hydriodide | 2863-34-5 | >98.00% | |
Bethanidine hydriodide is an orally active antihypertensive agent and adrenergic neuron blocker. | ||||
| GC90924 | TNP-GTP (sodium salt) | - | >95.00% | |
مشتق فلورسنت لـ GTP | ||||
| GC90952 | 1-Aminoguanosine-3',5'-monophosphate (sodium salt) | 1380911-23-8 | >95.00% | |
مادة أساسية لإنزيم بروتين كيناز الـ cGMP-المعتمد. | ||||
| GC91090 | Oxamyl-d6 | 2470229-60-6 | >99.00% | |
معيار داخلي لتحديد كمية الأوكساميل | ||||
| GC91093 | MR2938 | 1044870-65-6 | >95.00% | |
مثبط للأستيل كولين استيراز (AChE) | ||||
| GC91114 | Xylazine-d6 (CRM) | 1228182-53-3 | - | |
مادة مرجعية معتمدة | ||||
| GC91180 | Carbofuran-d3 | 1007459-98-4 | >99.00% | |
معيار داخلي لتحديد كمية الكاربوفوران | ||||
| GC91181 | Malathion-d10 | 347841-48-9 | >99.00% | |
معيار داخلي لتحديد كمية المالاثيون | ||||
| GC91188 | Acephate-d3 | 2140327-70-2 | >99.00% | |
معيار داخلي لتحديد كمية الأسفات. | ||||
| GC91190 | Propoxur-d3 | 1219798-56-7 | >99.00% | |
معيار داخلي لتحديد كمية بروبوكسور | ||||
| GC92078 | PKG Inhibitor (trifluoroacetate salt) | - | >95.00% | |
PKG Inhibitor (trifluoroacetate salt) هو مثبط يعتمد على cGMP PKG Ki = 86 ميكرومتر. | ||||
| GN10069 | Ginsenoside Ro | 34367-04-9 | >98.00% | |
| GN10104 | Gramine | 87-52-5 | >98.00% | |