GLPBio

GPCR/G protein

Research Areas

Products Related to GPCR/G protein(3538)

  • GC80865 structure
    GC80865Anandamide- 15 N
    Purity: >99.50%

    Anandamide - 15 N (AEA- 15 N) is the 15 N-labeled Anandamide.

  • GC81037 structure
    GC81037AP-7-168
    CAS: 2816062-15-2
    Purity: >99.50%

    AP-7-168, molecular glues, is a β-arrestin-biased negative allosteric modulator of the β2-adrenergic receptor ( β2AR ).

  • GC81402 structure
    GC81402Sp-ATPαS tetrasodium solution (100mM)
    Purity: >98.50%

    Sp-ATPαS tetrasodium is a thiophosphonate analogue of ATP.

  • GC81433 structure
    GC81433PEN (human) TFA
    Purity: >97.00%

    PEN (human) TFA, one of the most abundant hypothalamic neuropeptide and derived from the proprotein ProSAAS, is an endogenous ligand of GPR83 [1] .

  • GC81434 structure
    GC81434RAS activator compound 1
    CAS: 1579978-17-8
    Purity: >98.50%

    RAS activator compound 1 (Compound 7c) is a RAS activator targeting the guanine nucleotide exchange factor (GEF) son of sevenless homologue 1 ( SOS1 ).

  • GC81435 structure
    GC814352-Bromo-LSD D-Tartrate
    CAS: 2855123-30-5
    Purity: >99.50%

    2-Bromo-LSD D-Tartrate (BOL-148 D-Tartrate) is a blood-brain barrier-permeable 5-HT 2A partial agonist and competitive partial antagonist.

  • GC81439 structure
    GC81439SZ0232
    CAS: 924851-91-2
    Purity: >99.00%

    SZ0232 is a selective mPGES-2 inhibitor.

  • GC81443 structure
    GC81443E8431
    CAS: 2419580-01-9
    Purity: >97.00%

    E8431 is a DCSTAMP antagonist with an IC 50 value of 775.8 nM for osteoclastogenesis.

  • GC81482 structure
    GC81482PF-07976016
    CAS: 3059496-70-4
    Purity: >98.00%

    PF-07976016 (GIPR antagonist 4) is an orally active GIPR antagonist with an IC 50 of 4.1 nM.

  • GC81496 structure
    GC81496TAVO101
    Purity: >96.50%

    TAVO101 is a humanized anti- TSLP antibody with an EC 50 of 0.19 nM against hTSLP.

  • GC81510 structure
    GC81510Denatonium benzoate-d 5
    Purity: >99.50%

    Denatonium benzoate -d 5 (THS-839-d 5 ) is the deuterium labeled Denatonium benzoate.

  • GC81558 structure
    GC81558ANT308 TFA
    Purity: >99.50%

    ANT308 TFA is a vasoactive intestinal polypeptide ( VIP receptor ) antagonist.

  • GC81559 structure
    GC81559Maxadilan TFA
    Purity: >96.00%

    Maxadilan TFA is a specific irreversible PAC1 receptor agonist and a potent vasodilator peptide present in the salivary glands of sand flies.

  • GC81560 structure
    GC81560GRK2 degrader-1
    CAS: 3052947-04-0
    Purity: >98.50%

    GRK2 degrader-1 (compound 1) is a potent and orally active GRK2 degrader.

  • GC81561 structure
    GC81561GR-11-1
    Purity: >98.50%

    GR-11-1 is a GRK2 substrate for phosphorylation.

  • GC81562 structure
    GC81562GUB08248 acetate
    Purity: >98.50%

    GUB08248 acetate is a full GPR10 agonist and a partial NPFF2R agonist, with EC 50 values of 0.5 nM and 2.5 nM, respectively.

  • GC81563 structure
    GC81563GUB10194 acetate
    Purity: >98.50%

    GUB10194 acetate is a fully potent and selective GPR10 agonist with an EC 50 of 15 nM.

  • GC81564 structure
    GC81564Z52
    CAS: 3077480-59-9
    Purity: >98.50%

    Z52 is a Ras protein inhibitor.

  • GC81565 structure
    GC81565palm11-PrRP31 TFA
    Purity: >99.00%

    palm11-PrRP31 TFA is a lipidized endogenous appetite inhibitory neuropeptide (PrRP) analogue.

  • GC81566 structure
    GC81566Ro 25-1553 TFA
    Purity: >99.00%

    Ro 25-1553 TFA is a 31 amino acid vasoactive intestinal peptide (VIP) analog, that acts as an agonist for VIP2 receptor ( VPAC2 receptor ).

  • GC81567 structure
    GC81567Ro 25-1553 acetate
    Purity: >98.00%

    Ro 25-1553 acetate is a selective VIP 2 receptor ( VPAC 2 receptor ) agonist.

  • GC81662 structure
    GC81662nor-MC3
    CAS: 2870681-06-2
    Purity: >98.00%

    nor-MC3 is an MC3 -type ionizable lipid with C 17 unsaturated chains, formulated in lipid nanoparticles for nucleic acid ( mRNA and siRNA) delivery and supports in vitro and in vivo transfection [1] .

  • GC81677 structure
    GC81677APJ receptor agonist 10 free base
    CAS: 2415197-87-2
    Purity: >99.00%

    APJ receptor agonist 10 free base is an agonist of the APJ Receptor.

  • GC81693 structure
    GC81693GPR52 agonist-4
    CAS: 1313195-88-8
    Purity: >98.00%

    GPR52 agonist-4 (Compound 65) is a highly selective G-protein-coupled receptor GPR52 modulator.