TP-472 |
| Catalog No.GC40628 |
Le TP-472 est un inhibiteur sélectif de BRD7/9, avec des KD de 0,34 μM et 33 nM pour BRD7 et BRD9, respectivement.
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Cas No.: 2079895-62-6
Sample solution is provided at 25 µL, 10mM.
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TP-472 is an inhibitor of bromodomain BRD9 (Kd = 33 nM; EC50 = 320 nM in a NanoBRET assay). It has >30-fold selectivity over all other bromodomain family members with the exception of the highly homologous BRD7 bromodomain (Kd = 340 nM in an isothermal titration calorimetry (ITC) assay). See the Structural Genomic Consortium (SGC) website for more information.
Average Rating: 5 (Based on Reviews and 26 reference(s) in Google Scholar.)
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