TP-472 |
Katalog-Nr.GC40628 |
TP-472 ist ein selektiver BRD7/9-Inhibitor mit KDs von 0,34 μM und 33 nM fÜr BRD7 bzw. BRD9.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 2079895-62-6
Sample solution is provided at 25 µL, 10mM.
TP-472 is an inhibitor of bromodomain BRD9 (Kd = 33 nM; EC50 = 320 nM in a NanoBRET assay). It has >30-fold selectivity over all other bromodomain family members with the exception of the highly homologous BRD7 bromodomain (Kd = 340 nM in an isothermal titration calorimetry (ITC) assay). See the Structural Genomic Consortium (SGC) website for more information.
Average Rating: 5
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