Tubulin inhibitor 6 (Synonyms: Improved Heterocyclic Activator of PP2A 1, Tubulin Inhibitor 6) |
Catalog No.GC39558 |
L'inhibiteur de tubuline 6 (composé 14b) est un inhibiteur de la tubuline et un puissant inhibiteur de plusieurs lignées cellulaires cancéreuses. L'inhibiteur de tubuline 6 inhibe la polymérisation de la tubuline avec une CI50 de 0,87 μM. L'inhibiteur de tubuline 6 inhibe la croissance des cellules K562 avec une IC50 de 840 nM.
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Cas No.: 105925-39-1
Sample solution is provided at 25 µL, 10mM.
Tubulin inhibitor 6 (Compound 14b) is a tubulin inhibitor and a potent inhibitor of multiple cancer cell lines. Tubulin inhibitor 6 inhibits tubulin polymerization with an IC50 of 0.87 μM. Tubulin inhibitor 6 inhibits K562 cell growth with an IC50 of 840 nM[1].
[1]. Prinz H, et al. N-benzoylated phenoxazines and phenothiazines: synthesis, antiproliferative activity, and inhibition of tubulin polymerization. J Med Chem. 2011 Jun 23;54(12):4247-63.
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