Acetyl-(D-Arg¹⁰,Cys¹¹,D-Phe¹⁴,Cys¹⁷)-β-MSH (10-17) amide |
| カタログ番号GA20520 |
非常に強力で選択的なβ-MSH由来のメラノコルチン4受容体（MC-4R）アゴニストで、サブナノモーラーの効力を持っています。人間のMC-4R、MC-1R、MC-3RおよびMC-5Rに対する結合親和性はそれぞれ0.55±0.06、16.78±1.53、56.79±4.66および<500 nMです。 H-6268を食事誘発性肥満ラットに14日間皮下注射したところ、脂肪量の減少効果が示されました。
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Cas No.: 819048-44-7
Sample solution is provided at 25 µL, 10mM.
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Highly potent and selective β-MSH-derived melanocortin-4 receptor (MC-4R) agonist with sub-nanomolar potency. The binding affinities for human MC-4R, MC-1R, MC-3R and MC-5R were 0.55 ± 0.06, 16.78 ± 1.53, 56.79 ± 4.66, and < 500 nM,
Average Rating: 5 (Based on Reviews and 22 reference(s) in Google Scholar.)
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