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LX7101 (hydrochloride)

カタログ番号GC44094

LX7101は、LIMキナーゼ(LIMK)1および2、Rho関連キナーゼ1(ROCK-1)、ROCK-2の強力な阻害剤であり、それぞれのIC50値は32、4.3、69、および32 nMです。

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LX7101 (hydrochloride) 化学構造

Cas No.: 2319882-48-7

サイズ 価格 在庫数 個数
1mg
$77.00
在庫あり
5mg
$308.00
在庫あり
10mg
$540.00
在庫あり

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Sample solution is provided at 25 µL, 10mM.

Description Chemical Properties Product Documents Related Products

LX7101 is a potent inhibitor of LIM kinase (LIMK) 1 and 2 and Rho-associated kinase 1 (ROCK-1) and ROCK-2 with IC50 values of 32, 4.3, 69, and 32 nM, respectively. It is selective, showing no cross reactivity in a panel of binding assays including 78 receptors and transporters and 430 additional kinases, at a concentration of 10 μM. Topical administration (3 μl of 1 mg/ml solution) of LX7101 to the eye reduces intraocular pressure in a dexamethasone-induced mouse model of glaucoma.

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Average Rating: 5 ★★★★★ (Based on Reviews and 32 reference(s) in Google Scholar.)

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