HSL-IN-1 |
カタログ番号GC36257 |
HSL-IN-1 (化合物 24b) は、強力で経口的に活性なホルモン感受性リパーゼ (HSL) 阻害剤 (IC50=2 nM) であり、反応性代謝物に対する感受性が大幅に低下しています 。
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Cas No.: 2095156-13-9
Sample solution is provided at 25 µL, 10mM.
HSL-IN-1 (compound 24b) is a potent and orally active hormone sensitive lipase (HSL) inhibitor (IC50=2 nM) with a significantly reduced reactive metabolite liability[1]. IC50: 2 nM (Hormone sensitive lipase)[1]
[1]. Ogiyama T, et al. Identification of a novel hormone sensitive lipase inhibitor with a reduced potential of reactive metabolites formation. Bioorg Med Chem. 2017 Apr 1;25(7):2234-2243.
Average Rating: 5
(Based on Reviews and 27 reference(s) in Google Scholar.)GLPBIO products are for RESEARCH USE ONLY. Please make sure your review or question is research based.
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