PROTAC ERRα ligand 2 |
| カタログ番号GC38383 |
PROTAC ERRαリガンド 2 は、5.67 nM の IC50 を持つエストロゲン関連受容体 α (ERRα) インバース アゴニストです。 PROTAC ERRαリガンド 2 (IC50=5.67 nM) は、XCT790 (IC50=61.3 nM) よりも約 11 倍改善された効力を示します。
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Cas No.: 2306388-57-6
Sample solution is provided at 25 µL, 10mM.
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PROTAC ERRα ligand 2 is an estrogen-related receptor α (ERRα) inverse agonist with an IC50 of 5.67 nM. PROTAC ERRα ligand 2 (IC50=5.67 nM) displays a ~11-fold improved potency than XCT790 (IC50=61.3 nM)[1].
[1]. Peng L, et al. Identification of New Small-Molecule Inducers of Estrogen-related Receptor α (ERRα) Degradation. ACS Med Chem Lett. 2019 Apr 12;10(5):767-772.
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