H4 Receptor antagonist 1 |
| カタログ番号GC31232 |
H4 受容体アンタゴニスト 1 は、強力で選択的なヒスタミン H4 受容体逆アゴニストであり、IC50 は 19 nM です。
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Cas No.: 848217-00-5
Sample solution is provided at 25 µL, 10mM.
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H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM.
H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM[1].
H4 Receptor antagonist 1 indicates that metabolic stability in rat microsomes is very low with only 1% parent compound remaining after 10 min incubation[1].
[1]. Cramp S, et al. Identification and hit-to-lead exploration of a novel series of histamine H4 receptor inverse agonists. Bioorg Med Chem Lett. 2010 Apr 15;20(8):2516-9.
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