SSTR5 antagonist 1 |
| カタログ番号GC65313 |
SSTR5 アンタゴニスト 1 は、hSSTR5 および mSSTR5 の IC50 がそれぞれ 9.6 および 57 nM である、強力で選択的な経口利用可能なソマトスタチン受容体サブタイプ 5 (SSTR5) アンタゴニストです。
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 1628741-91-2
Sample solution is provided at 25 µL, 10mM.
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SSTR5 antagonist 1 is a potent, selective, and orally available somatostatin receptor subtype 5 (SSTR5) antagonist with IC50s of 9.6 and 57 nM for hSSTR5 and mSSTR5, respectively. (Compound 25a)[1]
[1]. Hirose H, et al. Discovery of novel 5-oxa-2,6-diazaspiro[3.4]oct-6-ene derivatives as potent, selective, and orally available somatostatin receptor subtype 5 (SSTR5) antagonists for treatment of type 2 diabetes mellitus. Bioorg Med Chem. 2017 Aug 1;25(15):4175-4193.
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