SSTR5 antagonist 1 |
| Katalog-Nr.GC65313 |
SSTR5-Antagonist 1 ist ein potenter, selektiver und oral verfÜgbarer Antagonist des Somatostatin-Rezeptor-Subtyps 5 (SSTR5) mit IC50-Werten von 9,6 und 57 nM fÜr hSSTR5 bzw. mSSTR5.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 1628741-91-2
Sample solution is provided at 25 µL, 10mM.
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SSTR5 antagonist 1 is a potent, selective, and orally available somatostatin receptor subtype 5 (SSTR5) antagonist with IC50s of 9.6 and 57 nM for hSSTR5 and mSSTR5, respectively. (Compound 25a)[1]
[1]. Hirose H, et al. Discovery of novel 5-oxa-2,6-diazaspiro[3.4]oct-6-ene derivatives as potent, selective, and orally available somatostatin receptor subtype 5 (SSTR5) antagonists for treatment of type 2 diabetes mellitus. Bioorg Med Chem. 2017 Aug 1;25(15):4175-4193.
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