BRD-IN-3 |
| Catalog No.GC35552 |
BRD-IN-3((R,R)-36n)은 IC50이 7nM인 매우 강력한 PCAF 브로모도메인(BRD) 억제제입니다. BRD-IN-3은 또한 GCN5 및 FALZ에 대한 활성을 나타냅니다.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 2351938-32-2
Sample solution is provided at 25 µL, 10mM.
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BRD-IN-3 ((R,R)-36n) is a highly potent PCAF bromodomain (BRD) inhibitor, with an IC50 of 7 nM. BRD-IN-3 also exhibits activity against GCN5 and FALZ[1]. IC50: PCAF BRD[1].
[1]. Huang L, et al. Discovery of Pyrrolo[3,2- d]pyrimidin-4-one Derivatives as a New Class of Potent and Cell-Active Inhibitors of P300/CBP-Associated Factor Bromodomain. J Med Chem. 2019 May 9;62(9):4526-4542.
Average Rating: 5 (Based on Reviews and 6 reference(s) in Google Scholar.)
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