PROTAC EZH2 Degrader-1 |
| Catalog No.GC65509 |
강력한 PROTAC EZH2 분해제인 PROTAC EZH2 분해기-1(화합물 150d)은 2.7 nM의 IC50으로 EZH2 메틸트랜스퍼라제 활성에 대한 억제 효과를 발휘합니다. EZH2는 많은 종양 형성 및 발달 과정에서 중요한 역할을 합니다.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 2641601-67-2
Sample solution is provided at 25 µL, 10mM.
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PROTAC EZH2 Degrader-1 (Compound 150d), a potent PROTAC EZH2 Degrader, exerts inhibitory effect on EZH2 methyltransferase activity with the IC50 of 2.7 nM. EZH2 plays an important role in many tumorigenesis and development processes[1].
[1]. Juan Xia, et al. Targeting Enhancer of Zeste Homolog 2 for the Treatment of Hematological Malignancies and Solid Tumors: Candidate Structure-Activity Relationships Insights and Evolution Prospects. J Med Chem. 2022 May 26;65(10):7016-7043.
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