GPCR/G protein
Research Areas
- Neuropeptide FF/AF Receptors(51)
- Neuropeptide S Receptor(3)
- GPBA Receptor(3)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- Formyl Peptide Receptors(11)
- 5-HT Receptor(414)
- Acetylcholine(28)
- Adenosine Deaminase(10)
- Adenosine Receptor(138)
- Adenosine Kinase(5)
- Adiponectin Receptor(3)
- Adrenergic Receptor(431)
- Adrenergic Transporters(5)
- Apelin Receptor(9)
- Angiotensin Receptor(117)
- Bombesin Receptors(23)
- Bradykinin Receptors(29)
- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(111)
- Calcimimetic Agent(2)
- CaSR(25)
- CCK1 Receptors(7)
- CCK2 Receptors(7)
- CCR(95)
- Chemokine Receptors(23)
- CRF1 Receptors(10)
- CRF2 Receptors(3)
- CXCR(93)
- CysLT1 receptor(1)
- Endothelin Receptor(53)
- EP1 Receptor(2)
- EP4 Receptor(2)
- ERRγ(1)
- ETA Receptors(5)
- ETB Receptors(5)
- Free Fatty Acid Receptors(16)
- Galanin Receptors(11)
- Ghrelin Receptors(11)
- GHSR(20)
- GIP Receptor(5)
- Glucagon Receptor(54)
- Glucocorticoid Receptor(94)
- GLUT1(1)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(12)
- GPR109A(4)
- GPR119(10)
- GPR120(9)
- GPR35(10)
- GPR44(1)
- GPR55(11)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(57)
- LPA Receptor(12)
- LPL Receptor(62)
- LTD4 Receptor(1)
- mGluR (123)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(57)
- Melatonin Receptors(23)
- Motilin Receptor(7)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(26)
- NK2 Receptors(7)
- NK3 Receptor(5)
- NOP Receptor(20)
- NPY Receptors(26)
- Orexin(3)
- Orphan 7-TM Receptors(6)
- OX Receptor(52)
- Oxytocin Receptors(22)
- P2Y Receptor(65)
- PACAP Receptors(7)
- PAF Receptors(7)
- Peptide Receptors(14)
- PGD2 Receptor(1)
- Prostaglandin Receptor(174)
- Prostanoid Receptors(25)
- Protease-Activated Receptors(9)
- RGS(2)
- S1P receptor(8)
- Secretin Receptors(1)
- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(43)
- Sigma Receptor(59)
- Vasopressin Receptor(34)
- 17,20-lyase(4)
- Ras(163)
- Urotensin-II Receptor(10)
- VIP Receptors(6)
- EBI2/GPR183(7)
- TSH Receptor(10)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(20)
- GPR84(10)
- Neuromedin U Receptors(2)
- Kisspeptin Receptor(6)
- CRFR(27)
- RGS Protein(5)
- Urotensin Receptor(7)
- Cholecystokinin Receptor(28)
- GPR139(4)
- mAChR(191)
- MCHR1 (GPR24)(16)
- Neurokinin Receptor(76)
- cGMP(27)
- GRK(3)
- GPR88(1)
- Amylin Receptor(3)
- Arrestin(8)
- Mas-related G-protein-coupled Receptor (MRGPR)(6)
- GCGR(7)
- GLP Receptor(16)
- Succinate Receptor 1(1)
- PTHR(2)
- Protease Activated Receptor (PAR)(6)
- Free Fatty Acid Receptor(5)
- Formyl Peptide Receptor (FPR)(3)
- Hydroxycarboxylic Acid Receptor (HCAR)(2)
- RXFP Receptor(2)
- Adhesion G Protein-coupled Receptors (AGPCRs)(1)
- Taste Receptor(1)
- GPR52(1)
Products Related to GPCR/G protein(3538)
- GC79312TRV0109101CAS: 1401027-29-9Purity: >98%
TRV0109101 is a μ-opioid peptide receptor (MOPR) selective agonist ( K D = 70 nM) with blood-brain barrier permeability.
- GC79313Alixorexton enantiomerCAS: 2648350-16-5Purity: >99.00%
Alixorexton (ALKS 2680) enantiomer is the enantiomer of Alixorexton.
- GC79314OctoclothepineCAS: 13448-22-1Purity: >99.50%
Octoclothepin (Clorotepine) is a D 2 dopamine receptor antagonist and 5-HT 2 serotonin receptor antagonist, with K i values of 0.67 nM, 0.57 nM, and 0.19 nM for the dopamine D 2, 5-HT 2A, and 5-HT 2C receptors, respectively.
- GC79316L-797591 hydrochlorideCAS: 3026641-74-4Purity: >99.50%
L-797591 hydrochloride is a selective sst 1 agonist.
- GC79317SSTR3 Agonist-1CAS: 3086695-73-7Purity: >98.00%
SSTR3 Agonist-1 (Compound EX 38) is an orally active SSTR3 agonist, with an EC 50 of 0.14 nM.
- GC79319R06039-641CAS: 2138444-75-2Purity: >98.50%
R06039-641 is a neuropeptide S receptor ( NPSR ) agonist with an EC 50 of 169 nM.
- GC79320R06039-691CAS: 2138445-51-7Purity: >99.50%
R06039-691 is a neuropeptide S receptor ( NPSR ) agonist with an EC 50 of 93 nM.
- GC79321MRS 2179 ammoniumPurity: >99.00%
MRS 2179 ammonium is a selective and competitive antagonist for P2Y1 receptor, with K B of 0.177 μM [1] .
- GC79322TP receptor antagonist-3CAS: 165537-72-4Purity: >99.50%
TP receptor antagonist-3 (compound 51280) is a potent thromboxane A2 prostanoid ( TP ) receptor with an IC 50 of 15.7 nM against Human TP.
- GC79323Terutroban sodiumCAS: 609340-89-8Purity: >98.00%
Terutroban (S-18886) sodium is a selective and orally active thromboxane-prostaglandin (TP) receptor antagonist with an IC 50 of 16.4 nM.
- GC79324HTL0039732CAS: 2639366-75-7Purity: >99.00%
HTL0039732 is an orally active antagonist of the prostaglandin EP4 receptor (Prostaglandin E2 Receptor EP4).
- GC79325ML161 analog 1CAS: 423740-83-4Purity: >99.50%
ML161 analog 1 (compound 38) is an analog of ML161.
- GC79326Tirzepatide sodiumPurity: >98.00%
Tirzepatide sodium (LY3298176 sodium) is a dual glucose-dependent insulinotropic polypeptide ( GIP ) and glucagon-like peptide-1 ( GLP-1 ) receptor agonist.
- GC79327BMS-986331CAS: 2375684-52-7Purity: >99.50%
BMS-986331 is an orally active selective N-Formyl Peptide Receptor 2 (FPR2) agonist with an EC 50 of 0.5 nM in humans and 1 nM in rats.
- GC79372Rosnilimab (Mouse IgG2a)Purity: >98.00%
Rosnilimab (Mouse IgG2a ) is a mouse-derived IgG2a antibody, Rosnilimab.
- GC79374PD-1/PD-L1-IN-63CAS: 2691796-92-4Purity: >98.00%
PD-1/PD-L1-IN-63 is an orally active PD-1/PD-L1 inhibitor with an IC 50 of 9.1 nM.
- GC79405TSLP modulator-1Purity: >99.50%
TSLP modulator-1 (Compound 14O) is a potent TSLP signaling modulator.
- GC79450Hydrocortisone-OVAPurity: >98%
Hydrocortisone -OVA is a conjugate of Hydrocortisone and OVA peptide.
- GC79504(R)-VerapamilCAS: 38321-02-7Purity: >98.50%
(R)-Verapamil (Dexverapamil) is an optically enantiomer of the oral-active Verapamil.
- GC79505RPI-GLYT2-82Purity: >99.00%
RPI-GLYT2-82 is a reversible, blood-brain barrier-permeable allosteric inhibitor of GlyT2 with an IC 50 value of 554 nM.
| Catalog No. | Product Name | CAS No. | Purity | Structure |
|---|---|---|---|---|
| GC79312 | TRV0109101 | 1401027-29-9 | >98% | |
TRV0109101 is a μ-opioid peptide receptor (MOPR) selective agonist ( K D = 70 nM) with blood-brain barrier permeability. | ||||
| GC79313 | Alixorexton enantiomer | 2648350-16-5 | >99.00% | |
Alixorexton (ALKS 2680) enantiomer is the enantiomer of Alixorexton. | ||||
| GC79314 | Octoclothepine | 13448-22-1 | >99.50% | |
Octoclothepin (Clorotepine) is a D 2 dopamine receptor antagonist and 5-HT 2 serotonin receptor antagonist, with K i values of 0.67 nM, 0.57 nM, and 0.19 nM for the dopamine D 2, 5-HT 2A, and 5-HT 2C receptors, respectively. | ||||
| GC79315 | VU6052254 | 3035701-02-8 | >98.00% | |
VU6052254, a derivative of VU0467319, is a selective, potent, orally active and brain-penetrant muscarinic M1 acetylcholine receptor ( mAChR1 ) positive allosteric modulator with an EC 50 of 59 nM. | ||||
| GC79316 | L-797591 hydrochloride | 3026641-74-4 | >99.50% | |
L-797591 hydrochloride is a selective sst 1 agonist. | ||||
| GC79317 | SSTR3 Agonist-1 | 3086695-73-7 | >98.00% | |
SSTR3 Agonist-1 (Compound EX 38) is an orally active SSTR3 agonist, with an EC 50 of 0.14 nM. | ||||
| GC79318 | NOTA-TATE | 709043-21-0 | >98.50% | |
NOTA-TATE is a somatostatin receptor 2 ( SSTR2 ) binder. | ||||
| GC79319 | R06039-641 | 2138444-75-2 | >98.50% | |
R06039-641 is a neuropeptide S receptor ( NPSR ) agonist with an EC 50 of 169 nM. | ||||
| GC79320 | R06039-691 | 2138445-51-7 | >99.50% | |
R06039-691 is a neuropeptide S receptor ( NPSR ) agonist with an EC 50 of 93 nM. | ||||
| GC79321 | MRS 2179 ammonium | - | >99.00% | |
MRS 2179 ammonium is a selective and competitive antagonist for P2Y1 receptor, with K B of 0.177 μM [1] . | ||||
| GC79322 | TP receptor antagonist-3 | 165537-72-4 | >99.50% | |
TP receptor antagonist-3 (compound 51280) is a potent thromboxane A2 prostanoid ( TP ) receptor with an IC 50 of 15.7 nM against Human TP. | ||||
| GC79323 | Terutroban sodium | 609340-89-8 | >98.00% | |
Terutroban (S-18886) sodium is a selective and orally active thromboxane-prostaglandin (TP) receptor antagonist with an IC 50 of 16.4 nM. | ||||
| GC79324 | HTL0039732 | 2639366-75-7 | >99.00% | |
HTL0039732 is an orally active antagonist of the prostaglandin EP4 receptor (Prostaglandin E2 Receptor EP4). | ||||
| GC79325 | ML161 analog 1 | 423740-83-4 | >99.50% | |
ML161 analog 1 (compound 38) is an analog of ML161. | ||||
| GC79326 | Tirzepatide sodium | - | >98.00% | |
Tirzepatide sodium (LY3298176 sodium) is a dual glucose-dependent insulinotropic polypeptide ( GIP ) and glucagon-like peptide-1 ( GLP-1 ) receptor agonist. | ||||
| GC79327 | BMS-986331 | 2375684-52-7 | >99.50% | |
BMS-986331 is an orally active selective N-Formyl Peptide Receptor 2 (FPR2) agonist with an EC 50 of 0.5 nM in humans and 1 nM in rats. | ||||
| GC79328 | HDB-1 | 3021527-82-9 | >98.00% | |
HDB-1 is a selective inhibitor of the P2Y14 receptor ( P2Y14R ) with an IC 50 of 26 pM. | ||||
| GC79372 | Rosnilimab (Mouse IgG2a) | - | >98.00% | |
Rosnilimab (Mouse IgG2a ) is a mouse-derived IgG2a antibody, Rosnilimab. | ||||
| GC79373 | FK3453 | 560111-91-3 | >99.50% | |
FK3453 is a dual adenosine A1/A2 inhibitor and a TSLP inhibitor. | ||||
| GC79374 | PD-1/PD-L1-IN-63 | 2691796-92-4 | >98.00% | |
PD-1/PD-L1-IN-63 is an orally active PD-1/PD-L1 inhibitor with an IC 50 of 9.1 nM. | ||||
| GC79405 | TSLP modulator-1 | - | >99.50% | |
TSLP modulator-1 (Compound 14O) is a potent TSLP signaling modulator. | ||||
| GC79450 | Hydrocortisone-OVA | - | >98% | |
Hydrocortisone -OVA is a conjugate of Hydrocortisone and OVA peptide. | ||||
| GC79504 | (R)-Verapamil | 38321-02-7 | >98.50% | |
(R)-Verapamil (Dexverapamil) is an optically enantiomer of the oral-active Verapamil. | ||||
| GC79505 | RPI-GLYT2-82 | - | >99.00% | |
RPI-GLYT2-82 is a reversible, blood-brain barrier-permeable allosteric inhibitor of GlyT2 with an IC 50 value of 554 nM. | ||||