- Bestell-Nr. Artikelname Informationen
- GC40105 βARK1 Inhibitor βARK1-Inhibitor (Methyl-5-[2-(5-nitro-2-furyl)vinyl]-2-furoat) ist ein GRK2 (β-ARK1)-Inhibitor.
- GC52006 CB-096 An inhibitor of RAN translation
- GC49117 Guanadrel Guanadrel ist ein oral aktiver postganglionÄrer adrenerger Inhibitor von Spiroketal.
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GC49089
FR900359
A cyclic depsipeptide and an inhibitor of Gαq, Gα11, and Gα14
- GC46233 Trandolaprilat (hydrate) Trandolaprilat (Hydrat) ist ein starker Hemmer des Angiotensin-Converting-Enzyms (ACE).
- GC45903 Quazinone A PDE3 inhibitor
- GC43803 HA-1077 (hydrochloride) Fasudil (HA-1077; AT877) dihydrochloride is a nonspecific RhoA/ROCK inhibitor and also has inhibitory effect on protein kinases, with an Ki of 0.33 μM for ROCK1, IC50s of 0.158 μM and 4.58 μM, 12.30 μ ;M, 1.650 μM fÜr ROCK2 bzw. PKA, PKC, PKG. HA-1077 (Hydrochlorid) ist auch ein potenter Ca2+-Kanalantagonist und Vasodilatator.
- GC43802 HA-1004 (hydrochloride) HA-1004 is an inhibitor of protein kinase G (PKG) and PKA (Kis = 1.4 and 2.3 μM, respectively).
- GC19438 TMB 8 (hydrochloride) TMB 8 is a non-competitive antagonist of nicotinic acetylcholine receptors (nAChRs) with IC50 values of 390 and 350 nM, respectively, for human muscle-type and α3β4 subunit-containing ganglionic nAChRs expressed in TE671/RD or SH-SY5Y cells.