MDR-652 |
| Katalog-Nr.GC39828 |
MDR-652 ist ein hochspezifischer und wirksamer transienter Rezeptorpotential-Vanilloid-1 (TRPV1)-Ligand mit agonistischer AktivitÄt.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 1933528-96-1
Sample solution is provided at 25 µL, 10mM.
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MDR-652 is a highly specific and efficacious transient receptor potential vanilloid 1 (TRPV1) ligand with agonist activity. The Kis are 11.4 and 23.8 nM for hTRPV1 and rTRPV1, respectively. The EC50s are 5.05 and 93 nM for hTRPV1 and rTRPV1, respectively. Potent topical analgesic activity[1].
[1]. Jihyae Ann, et al. Discovery of Nonpungent Transient Receptor Potential Vanilloid 1 (TRPV1) Agonist as Strong Topical Analgesic. J Med Chem. 2020 Jan 9;63(1):418-424.
Average Rating: 5 (Based on Reviews and 17 reference(s) in Google Scholar.)
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