AMG 333 |
カタログ番号GC65611 |
AMG 333 は、強力で選択性の高い TRPM8 アンタゴニストであり、IC50 は 13 nM です。
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Cas No.: 1416799-28-4
Sample solution is provided at 25 µL, 10mM.
AMG 333 is a potent and highly selective TRPM8 antagonist with an IC50 of 13 nM.
[1]. Horne DB, et al. Discovery of TRPM8 Antagonist ( S)-6-(((3-Fluoro-4-(trifluoromethoxy)phenyl)(3-fluoropyridin-2-yl)methyl)carbamoyl)nicotinic Acid (AMG 333), a Clinical Candidate for the Treatment of Migraine. J Med Chem. 2018 Sep 27;61(18):8186-8201.
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