Snail/HDAC-IN-1 |
カタログ番号GC69917 |
Snail/HDAC-IN-1は、効果的なSnail/HDAC二重標的阻害剤です。Snail/HDAC-IN-1は、HDAC1に対して強力な抑制活性を示し、IC50値は0.405μMであり、またSnailに対しても強力な抑制作用を示し、Kd値は0.18μMです。Snail/HDAC-IN-1はHCT-116細胞中のヒストンH4アセチル化を増加させ、同時にSnailタンパク質の発現を低下させるため、細胞凋亡(アポトーシス)を誘導します。
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 2415281-52-4
Sample solution is provided at 25 µL, 10mM.
Review for Snail/HDAC-IN-1
Average Rating: 5
(Based on Reviews and 30 reference(s) in Google Scholar.)Review for Snail/HDAC-IN-1
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