GSK8573 |
| Catalog No.GC38049 |
GSK8573은 GSK2801(BAZ2A 및 BAZ2B 브로모도메인의 아세틸-리신 경쟁 억제제)에 대한 비활성 대조군 화합물입니다. GSK8573은 1.04μM의 Kd 값으로 BRD9에 대한 결합 활성을 가지며 BAZ2A/B 및 기타 브로모도메인 패밀리에 대해 비활성입니다. GSK8573은 생물학적 실험에서 구조적으로 관련된 음성 대조군 화합물로 사용될 수 있습니다.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 1693766-04-9
Sample solution is provided at 25 µL, 10mM.
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GSK8573 (compound 23) is an inactive control compound for GSK2801. GSK8573 has binding activity to BRD9 with a Kd value of 1.04 μM and is inactive against BAZ2A/B and other bromodomain familiy[1].
[1]. Chen P, et al. Discovery and Characterization of GSK2801, a Selective Chemical Probe for the Bromodomains BAZ2A and BAZ2B. J Med Chem. 2016 Feb 25;59(4):1410-24.
Average Rating: 5 (Based on Reviews and 31 reference(s) in Google Scholar.)
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