LSD1-IN-7 benzenesulfonate (Synonyms: CC-90011 benzenesulfonate; LSD1-IN-7 benzenesulfonate) |
| Catalog No.GC39287 |
CC-90011 벤젠술포네이트는 IC50이 0.25nM인 라이신 특이적 데메틸라제-1(LSD1)의 강력하고 선택적이고 가역적이며 경구 활성 억제제입니다. CC-90011 벤젠술포네이트는 LSD2, MOA-A 및 MAO-B에 대한 효소 억제가 적습니다. CC-90011 벤젠술포네이트는 급성 골수성 백혈병(AML) 및 소세포 폐암(SCLC) 세포 분화를 유도하고 강력한 항암 활성을 가지고 있습니다.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 2097523-60-7
Sample solution is provided at 25 µL, 10mM.
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LSD1-IN-7 benzenesulfonate is a potent and orally active inhibitor of lysine specific demethylase-1 (LSD1) with anticancer activity extracted from patent WO2017079670A1, compound 4-[2-(4-amino-piperidin-1-yl)-5-(3-fluoro-4-methoxy-phenyl)-1-methyl-6-oxo-1,6-dihydro-pyrimidin-4-yl]-2-fluorobenzonitrile[1].
[1]. Young K. Chen, et al. Compositions comprising an inhibitor of lysine specific demethylase-1. WO2017079670A1.
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