8-Cyclopentyl-1,3-dimethylxanthine (Synonyms: CPT, 8-Cyclopentyltheophylline, NSC 101806) |
| Katalog-Nr.GC50354 |
8-Cyclopentyl-1,3-dimethylxanthin (Verbindung 2a) ist ein selektiver Adenosin-A1-Rezeptorantagonist mit Kis von 10,9 nM und 1440 nM fÜr den A1-Rezeptor bzw. den A2-Rezeptor.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 35873-49-5
Sample solution is provided at 25 µL, 10mM.
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High affinity adenosine A1 receptor antagonist (pKi = 7.5-8).
Dalpiaz et al (1998) Thermodynamics of full agonist, partial agonist, and antagonist binding to wild-type and mutant adenosine A1 receptors. Biochem.Pharmacol. 56 1437 PMID:9827575
Average Rating: 5 (Based on Reviews and 38 reference(s) in Google Scholar.)
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