AGI-24512 |
Katalog-Nr.GC33019 |
AGI-24512 ist ein potenter Hemmer der Methioninadenosyltransferase 2α (MAT2A) mit einem IC50 von 8 nM. AGI-24512 lÖst eine DNA-Schadensreaktion aus. AGI-24512 kann die Proliferation von MTAP-deletierten Krebszellen in vitro blockieren. AGI-24512 kann fÜr die Erforschung von Krebserkrankungen verwendet werden.
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Cas No.: 2201066-53-5
Sample solution is provided at 25 µL, 10mM.
AGI-24512 is a methionine adenosyltransferase 2A (MATA2 ) inhibitors useful for treatment of cancer. AGI-24512 blocks growth of MTAP-deleted cancer cells in vitro.
[1]. Agios. Targeting MAT2A in MTAP-deleted Cancers. Presented at the American Association for Cancer Research (AACR) Annual Meeting, April 14-18, 2018, Chicago, IL, USA
Average Rating: 5
(Based on Reviews and 17 reference(s) in Google Scholar.)GLPBIO products are for RESEARCH USE ONLY. Please make sure your review or question is research based.
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