CTAP TFA |
| カタログ番号GC60730 |
CTAP TFA は、IC50 が 3.5 nM の、強力で選択性の高い BBB 浸透性の μ オピオイド受容体アンタゴニストです。
Products are for research use only. Not for human use. We do not sell to patients.
Sample solution is provided at 25 µL, 10mM.
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CTAP TFA is a potent, highly selective, and brain penetrant μ opioid receptor antagonist (IC50=3.5 nM) and displays over 1200-fold selectivity over δ opioid (IC50=4500 nM) and somatostatin receptors. CTAP TFA can be used for the study of L-DOPA-induced dyskinesia (LID)[1].
[1]. Mitchell J Bartlett, et al. Highly-selective µ-opioid Receptor Antagonism Does Not Block L-DOPA-induced Dyskinesia in a Rodent Model.BMC Res Notes
Average Rating: 5 (Based on Reviews and 18 reference(s) in Google Scholar.)
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