GR 103691 |
| カタログ番号GC38022 |
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 162408-66-4
Sample solution is provided at 25 µL, 10mM.
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GR 103691 is a potent, selective dopamine D3 receptor antagonist with a Ki value of 0.4 nM. GR 103691 shows more than 100-fold selectivity for human dopamine human (h)D3 over hD4 and hD1 sites[1].
GR 103691 shows marked affinity for serotonin1A (5-HT1A) receptors (Ki of 5.8 nM) and α-1 adrenoceptors (Ki of 12.6 nM)[1].
[1]. Audinot V, et al. A comparative in vitro and in vivo pharmacological characterization of the novel dopamine D3 receptor antagonists (+)-S 14297, nafadotride, GR 103,691 and U 99194. J Pharmacol Exp Ther. 1998 Oct;287(1):187-97.
Average Rating: 5 (Based on Reviews and 37 reference(s) in Google Scholar.)
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