Perphenazine (Synonyms: NSC 150866, SCH 3940) |
| カタログ番号GC12293 |
ペルフェナジンは経口活性ドーパミン受容体およびヒスタミン 1 受容体アンタゴニストであり、Ki 値はそれぞれ 0.56 nM (D2)、0.43 nM (D3)、6 nM (5-HT2A) です。
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Cas No.: 58-39-9
Sample solution is provided at 25 µL, 10mM.
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Perphenazine is a typical antipsychotic drug, inhibits 5-HT2Areceptor, Alpha-1A adrenergic receptor, Dopamine receptor D2/D3, D2L receptor, and Histamine H1 receptor, with Ki values of 5.6, 10, 0.765/0.13, 3.4, and 8 nM, respectively.
References:
[1]. Richtand NM, et al. Dopamine and serotonin receptor binding and antipsychotic efficacy. Neuropsychopharmacology. 2007 Aug;32(8):1715-26.
Average Rating: 5 (Based on Reviews and 33 reference(s) in Google Scholar.)
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