GR 159897 |
| Katalog-Nr.GC16408 |
GR 159897 ist ein hochwirksamer, selektiver, kompetitiver, nicht-peptidischer Neurokinin 2 (NK2)-Rezeptorantagonist, der in das Gehirn eindringt.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 158848-32-9
Sample solution is provided at 25 µL, 10mM.
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GR 159897 is a highly potent, selective, competitive, brain-penetrated non-peptide antagonist at tachykinin NK2 receptors, inhibits binding of [3H]GR100679 to hNK2-CHO cells and rat colon membranes with pKis of 9.51 and 10, respectively. Antagonizes bronchoconstriction, with anxiolytic-like activity[1].
References:
[1]. Beresford IJ, et al. GR159897, a potent non-peptide antagonist at tachykinin NK2 receptors. Eur J Pharmacol. 1995 Jan 16;272(2-3):241-8.
Average Rating: 5 (Based on Reviews and 35 reference(s) in Google Scholar.)
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