GSK4028 |
| Katalog-Nr.GC30714 |
GSK4028 ist die enantiomere Negativkontrolle von GSK4027, einer chemischen PCAF/GCN5-BromodomÄnensonde, der pIC50 von GSK4028 betrÄgt 4,9 in einem zeitaufgelÖsten Fluoreszenzresonanzenergietransfer (TR-FRET)-Assay.
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Cas No.: 2079886-19-2
Sample solution is provided at 25 µL, 10mM.
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GSK4028 is the enantiomeric negative control of GSK4027, which is a PCAF/GCN5 bromodomain chemical probe, the pIC50 of GSK4028 is 4.9 in a time-resolved fluorescence resonance energy transfer (TR-FRET) assay.
GSK4028 is the enantiomeric negative control of GSK4027, which is a PCAF/GCN5 bromodomain chemical probe, the pIC50 of GSK4028 is 4.9. GSK4028 also demonstrates potency toward BRD4 BD1 and BRD9 inTR-FRET assay with pIC50s of <4.3 and 4.5±0.13, respectively[1].
[1]. Humphreys PG, et al. Discovery of a Potent, Cell Penetrant, and Selective p300/CBP-Associated Factor (PCAF)/General Control Nonderepressible 5 (GCN5) Bromodomain Chemical Probe. J Med Chem. 2017 Jan 26;60(2):695-709.
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