Terodiline hydrochloride |
Catalog No.GC39186 |
테로딜린 염산염은 토끼 정관(M1), 심방(M2), 방광(M3) 및 회장 근육(M3)에서 각각 15, 160, 280 및 198nM의 Kbs를 갖는 M1 선택적 무스카린 수용체(mAChR) 길항제입니다. .
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 7082-21-5
Sample solution is provided at 25 µL, 10mM.
Terodiline hydrochloride is an M1-selective muscarinic receptor (mAChR) antagonist with Kbs of 15, 160, 280, and 198 nM in rabbit vas deferens (M1), atria (M2), bladder (M3) and ileal muscle (M3), respectively. Terodiline hydrochloride also is a Ca2+ blocker. Terodiline hydrochloride acts as a treatment for urinary frequency and urge incontinence[1].
[1]. Noronha-Blob L, et al. (+/-)-Terodiline: an M1-selective muscarinic receptor antagonist. In vivo effects at muscarinic receptors mediating urinary bladder contraction, mydriasis and salivary secretion. Eur J Pharmacol. 1991 Aug 29;201(2-3):135-42.
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