Neuroscience
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Neuroscience
Neurons communicate with each other, effector organs and sensory organs through the neurotransmitter – receptor pathway at synapses. Neurotransmitters can be divided into 4 major groups: 1. Amino acids (glumate, aspartate, serine, glycine and GABA); 2. Monoamines (norepinephrine, epinephrine, dopamine, histamine, and serotonin); 3. Peptides (opioid peptides, substance P, somatostatin); and 4. Others (acetylcholine, NO, nucleosides).
Targets for Neuroscience
- 5-HT Receptor(510)
- AChR(57)
- AChE(103)
- Alzheimer(88)
- Amyloid β(130)
- BACE(5)
- CGRP (29)
- COX(286)
- DAPK(5)
- Dopamine Receptor(295)
- GABA Receptor(225)
- Gap Junction(15)
- GluR(121)
- Histamine(2)
- Histamine Receptor(229)
- mPEGS-1(4)
- Muscarinic Receptor(42)
- Neuroscience Peptides(47)
- Nicotinic Receptor(65)
- P2 Receptor(2)
- P2X7 receptor(3)
- SSRIs(7)
- Substance P/NK1 Receptor(20)
- NMDA(2)
- Cholecystokinin Receptor(22)
- GPR139(3)
- mAChR(132)
- MCHR1 (GPR24)(15)
- Neurokinin Receptor(58)
- iGluR(130)
- nAChR(60)
- Beta-secretase(24)
- CaMK(28)
- Dopamine Transporter(17)
- Monoamine Oxidase(78)
- Serotonin Transporter(54)
- Behavioral Neuroscience(274)
- DREADD(0)
- Huntington(10)
- Neuroendocrinology(39)
- Neuroprotection(81)
- Ophthalmology(116)
- Pain Research(166)
- Parkinson(49)
- Seizure Disorders(74)
- Prion(6)
- Cholinesterases(13)
Products for Neuroscience
- Cat.No. Nombre del producto Información
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GC63267
α-Chaconine
La α-chaconina inhibe las expresiones de COX-2, IL-1β, IL-6 y TNF-α a nivel transcripcional.
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GC49097
α-Conotoxin AuIB (trifluoroacetate salt)
GCCSYPPCFATNPDC
A conotoxin and an antagonist of α3β4 subunit-containing nAChRs -
GC26093
α-Conotoxin GI
α-Conotoxin GI, a 13-residue peptide originally isolated from the venom of the fish-hunting cone snail Conus geographus, acts as a competitive antagonist for the muscle-type nicotinic acetylcholine receptor (nAChR) with excellent selectivity for α/δ receptor subunit binding over α/γ.
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GC49140
α-Conotoxin ImI (trifluoroacetate salt)
α-CTx ImI, GCCSDPRCAWRC
A conotoxin and an antagonist of α7 nAChRs -
GC49838
α-Cortolone
20α-Cortolone, NSC 59872
A metabolite of cortisol -
GC40262
α-Humulene
αCaryophyllene, (±)-αHumulene
α-El humuleno es un constituyente principal de Tanacetum vulgare L. -
GC64563
α-Methylserotonin
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GC48292
α-MSH (human, mouse, rat, porcine, bovine, ovine) (trifluoroacetate salt)
α-Melanocyte-stimulating Hormone, Ac-SYSMEHFRWGKPV-NH2
α-MSH (α-Melanocyte-Stimulating Hormone) TFA, un neuropéptido endÓgeno, es un agonista endÓgeno del receptor 4 de melanocortina (MC4R) con actividades antiinflamatorias y antipiréticas. -
GC41499
α-Phellandrene
p-Mentha-1,5-diene, (±)-α-Phellandrene
α-Phellandrene is a cyclic monoterpene that has been found in various plants, including Cannabis, and has diverse biological activities. -
GC10873
α-Spinasterol
Bessisterol, Hitodesterol
α-La espinasterol, aislada de Spinacia oleracea, tiene actividad antibacteriana. -
GC63615
α-Thujone
α-La tujona es un monoterpeno aislado del aceite esencial de Thuja occidentalis con potentes actividades antitumorales.
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GC70179
α7 Nicotinic receptor agonist-1
α7 Agonista del receptor nicotínico-1 (Preparación 5) es un agonista del receptor nAChR α7. El Agonista del receptor nicotínico-1 α7 se puede utilizar en trastornos psiquiátricos (como la esquizofrenia, el trastorno bipolar o depresión maníaca y la ansiedad) y discapacidades intelectuales (como la enfermedad de Alzheimer, los déficits de aprendizaje, los déficits cognitivos, el trastorno por déficit de atención e hiperactividad, pérdida de memoria y demencia con cuerpos de Lewy) para investigación.
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GC49467
β-Aescin
A triterpenoid saponin with diverse biological activities
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GC63273
β-Amyloid (1-14),mouse,rat
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GC66089
β-Amyloid (1-40) (TFA)
Amyloid Beta-Peptide (1-40) (human) TFA; Amyloid β-Peptide (1-40) (human) TFA
β-Amyloid (1-40) TFA es una proteÍna primaria en las placas que se encuentran en los cerebros de pacientes con la enfermedad de Alzheimer's. -
GC70182
β-Amyloid (1-40), FAM-labeled TFA
β-Amiloide (1-40), TFA marcado con FAM, es un péptido de β-amiloide (1-40) marcado con fluorescencia FAM (Λex= 492 nm y Λem= 518 nm).
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GC63274
β-Amyloid (1-42), (rat/mouse) (TFA)
Amyloid β-peptide (1-42) (rat/mouse) TFA
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GC37984
β-Amyloid (1-42), rat
Amyloid β-peptide (1-42) (rat/mouse)
β-amiloide (1-42), la rata es un péptido de 42 aa, muestra un efecto citotÓxico en cortes agudos del hipocampo y se utiliza en la investigaciÓn de la enfermedad de Alzheimer's. -
GC66416
β-Amyloid (22-35) (TFA)
Amyloid β-Protein (22-35) (TFA)
β-Amyloid 22-35 (Amyloid β-Protein 22-35) TFA, el fragmento de residuos 22-35 de β-proteÍna amiloide, tiene un efecto citotÓxico en neuronas cultivadas del hipocampo de rata en medio sin suero. β-Amyloid 22-35 TFA forma agregados y fibrillas amiloides tÍpicas que se asemejan a las de la β-proteÍna amiloide en soluciÓn tampÓn neutra). -
GC66346
β-Amyloid (42-1), human TFA
Amyloid β Peptide (42-1)(human) TFA
β-amiloide (42-1), TFA humano es la forma inactiva de amiloide β Péptido (1-42). β-Amyloid (42-1), TFA humano es un péptido de 42 aminoÁcidos que juega un papel clave en la patogénesis de la enfermedad de Alzheimer. -
GC37986
β-Amyloid 1-17
β-Amyloid 1-17 es un péptido de β-amiloide, estabiliza las fibras y juega un papel en la formación de fibras Aβ.
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GC37987
β-Amyloid 1-20
β-Amyloid 1-20 consta de los aminoácidos 1 a 20 de la proteína beta amiloide.
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GC37993
β-Amyloid 1-9
β-Amyloid 1-9, un fragmento N-terminal de beta amiloide, consta de los residuos de aminoácidos 1 a 9.
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GC37985
β-Amyloid 11-22
β-Amyloid 11-22 es un fragmento peptídico de β-amiloide.
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GC37988
β-Amyloid 12-20
β-Amyloid 12-20 es un fragmento peptídico de β-amiloide.
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GC37991
β-Amyloid 15-21
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GC37992
β-Amyloid 18-28
β-Amyloid 18-28 es un fragmento peptídico de β-amiloide.
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GC37994
β-Amyloid 22-40
β-Amyloid 22-40 es un fragmento peptídico de β-amiloide.
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GC37995
β-Amyloid 33-40
β-Amyloid 33-40 es un péptido que consiste en el aminoácido 33 a 40 de la proteína beta amiloide.
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GC37996
β-Amyloid 35-42
β-Amyloid 35-42 es un péptido que consiste en el aminoácido 35 a 42 de la proteína beta amiloide.
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GC37997
β-Amyloid 4-10
β-Amyloid 4-10 es un epítopo para el anticuerpo policlonal anti-Aβ(1-42), reduce la deposición de amiloide en un modelo de ratón transgénico con enfermedad de Alzheimer.
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GC34944
β-CGRP, human TFA
Human β-CGRP TFA; CGRP-II (Human) (TFA)
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GC41623
β-Elemonic Acid
Elemadienonic Acid, 3-Oxotirucallenoic Acid, 3-oxo Tirucallic Acid
β-El Ácido elemÓnico es un triterpeno aislado de Boswellia papyrifera. -
GC45234
β-Endorphin (1-27) (human) (trifluoroacetate salt)
β-Endorphin (1-27) is an endogenous peptide that binds to μ-, δ-, and κ-opioid receptors (Kis = 5.31, 6.17, and 39.82 nM, respectively, in COS-1 cells expressing rat receptors).
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GC45236
β-Endorphin (rat)
β-Endorphin (β-EP) is an endogenous opioid neuropeptide with diverse biological activities.
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GC52494
β-Endorphin (rat) (trifluoroacetate salt)
An opioid neuropeptide
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GC49769
β-Glucogallin
1-O-Galloyl-β-D-glucose
A plant metabolite and an aldose reductase 2 inhibitor -
GC40105
βARK1 Inhibitor
βInhibidor de ARK1 (5-[2-(5-nitro-2-furil)vinil]-2-furoato de metilo) es un inhibidor de GRK2 (β-ARK1).
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GC38010
γ-Aminobutyric acid
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GC64508
γ-Aminobutyric acid-d6
El ácido γ-aminobutírico-d6 (ácido 4-aminobutírico-d6) es el ácido γ-aminobutírico etiquetado con deuterio.
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GC49865
γ-D-Glutamylglycine (trifluoroacetate salt)
γ-DGG
An excitatory amino acid antagonist -
GC48313
γ-Lindane
An insecticide and GABAA receptor antagonist
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GC10872
α-Conotoxin AuIB
α-Conotoxin AuIB, a potent and selective α3β4 nicotinic acetylcholine receptor (nAChR) antagonist, blocks α3β4 nAChRs expressed in Xenopus oocytes with an IC50 of 0.75 μM.
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GC13644
α-Conotoxin EI
Selective antagonist of neuromuscular nicotinic receptors α1β1γδ
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GC14353
α-Conotoxin ImI
Nicotinic receptor antagonist
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GC14296
α-Conotoxin PIA
α-Conotoxin PIA es un antagonista del receptor nicotÍnico de acetilcolina (nAChR) que se dirige a los subtipos de nAChR que contienen las subunidades α6 y α3.
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GC10368
α-Conotoxin PnIA
α-Conotoxin PnIA, un antagonista potente y selectivo del α7 nAChR de mamÍferos, tiene potencial para la investigaciÓn de afecciones neurolÓgicas como el dolor neuropÁtico y la enfermedad de Alzheimer's.
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GC11577
α-Methyl-5-hydroxytryptamine maleate
α-Me-5-HT, α-Methyl-5-HT, α-Methyl-5-hydroxytryptamine, α-Methylserotonin
5-HT2B receptor agonist -
GC34242
β-Amyloid (1-42), rat TFA
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GC31146
β-Amyloid (10-35), amide
β-amiloide (10-35), la amida se compone de 26 aa (10-35 residuos del péptido Aβ) y es el componente principal de las placas amiloides de la enfermedad de Alzheimer.
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GC31129
β-Amyloid 1-16 (Amyloid β-Protein (1-16))
Amyloid β-Protein (1-16)
β-Amyloid 1-16 (Amyloid β-Protein (1-16)) es un fragmento de proteÍna β-Amyloid involucrado en la uniÓn de metales. -
GC31171
β-Amyloid 1-28 (Amyloid β-Protein (1-28))
Amyloid β-Protein (1-28)
β-Amyloid 1-28 (Amyloid β-Protein (1-28)) es un fragmento de proteÍna β-Amyloid involucrado en la uniÓn de metales. -
GC30325
β-Amyloid 22-35 (Amyloid β-Protein (22-35))
β-Amyloid 22-35 (Amyloid β-Protein 22-35), el fragmento de residuos 22-35 de β-proteÍna amiloide, tiene un efecto citotÓxico en neuronas cultivadas del hipocampo de rata en medio sin suero.
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GC31137
β-Amyloid 29-40 (Amyloid beta-protein(29-40))
β-amiloide 29-40 (proteÍna beta amiloide (29-40)) es un fragmento de amiloide-β péptido
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GC31179
β-Amyloid 31-35
β-Amyloid 31-35 es la secuencia más corta del péptido amiloide-β nativo que retiene la actividad neurotóxica.
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GC11449
β-CCB
benzodiazepine receptor ligand
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GC33595
β-CGRP, human (Human β-CGRP)
β-CGRP humano (Human β-CGRP) es uno de los péptidos calcitonina, actúa a través del complejo receptor similar a la calcitonina (CRLR) y proteína moduladora de actividad del receptor (RAMP), con IC50s de 1 nM y 300 nM para CRLR/RAMP1 y CRLR/RAMP2 en células.
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GC18033
γDGG
γDGG es un bloqueador competitivo del receptor AMPA.
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GC52013
(±)-10-hydroxy-12(Z)-Octadecenoic Acid
10-hydroxy-cis-12-Octadecenoic Acid
An oxylipin and metabolite of linoleic acid -
GC52421
(±)-10-hydroxy-12(Z)-Octadecenoic Acid-d5
10-hydroxy-cis-12-Octadecenoic Acid-d5
An internal standard for the quantification of (±)-10-hydroxy-12(Z)-octadecenoic acid -
GC41657
(±)-2-Amino-6,7-dihydroxy-1,2,3,4-tetrahydronaphthalene (hydrobromide)
(±)-ADTN, 6,7-ADTN, 6,7-diOHATN, NSC 287353
(±)-2-Amino-6,7-dihydroxy-1,2,3,4-tetrahydronaphthalene (6,7-ADTN) is a dopamine receptor agonist (EC50s = 3.5 and 0.65 μM in rat striatal and nucleus accumbens homogenates, respectively). -
GC41658
(±)-2-hydroxy Ibuprofen
(±)-2-hidroxi ibuprofeno es un metabolito de ibuprofeno.
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GC62726
(±)-Amiflamine
(±)-amiflamina (FLA 336) es un potente inhibidor de la monoaminooxidasa-A (MAO-A) con un pIC50 de 5,57.
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GC46272
(±)-Asenapine-13C-d3 (hydrochloride)
An internal standard for the quantification of (±)-asenapine
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GC46274
(±)-Baclofen-d4
(±)-Baclofen-d4 es el deuterio etiquetado como Baclofen.
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GC60394
(±)-Duloxetine hydrochloride
(Rac)-Duloxetine hydrochloride
El clorhidrato de (±)-duloxetina ((Rac)-duloxetina) es el racemato del clorhidrato de duloxetina. -
GC14410
(±)-Epibatidine
CMI 545
nicotinic agonist -
GC46288
(±)-Epibatidine (hydrochloride)
CMI 545 dihydrochloride
An agonist of α4β2 subunit-containing nAChRs -
GC46290
(±)-Ibuprofen-d3
DL-Ibuprofen-d3
El ibuprofeno D3 es un ibuprofeno etiquetado con deuterio. -
GC49515
(±)-Ibuprofen-d3 (sodium salt)
DL-Ibuprofen-d3
An internal standard for the quantification of (±)-ibuprofen -
GC45278
(±)-Ketoprofen-d3
(R,S)-Ketoprofen-d3, 2-(3-benzoylphenyl)Propionic Acid-d3
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GC12699
(±)-LY 395756
ligand for mGlu2 and mGlu3 receptor
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GC16735
(±)-McN 5652
5-HT uptake inhibitor
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GC49875
(±)-N-desmethyl Venlafaxine (hydrochloride)
Wy 45494
A minor active metabolite of venlafaxine -
GC46305
(±)-Nicotine-d3
DL-Nicotine-d3, (±)-Nicotine-methyl-d3
An internal standard for the quantification of (±)-nicotine -
GC14834
(±)-Nipecotic acid
(±)-Nipecotic Acid, (R,S)-Nipecotic Acid, 3-Piperidine Carboxylic Acid, DL-Piperidine 3-Carboxylic Acid
GABA uptake inhibitor -
GC41676
(±)-Nornicotine
DL-Nornicotine, (R,S)-Nornicotine
(±)-Nornicotine is a metabolite of nicotine that acts as a neuronal nicotinic acetylcholine receptor (nAChR) agonist. -
GC49482
(±)-Nornicotine-d4
DL-Nornicotine-d4, (R,S)-Nornicotine-d4
An internal standard for the quantification of (±)-nornicotine -
GC12394
(±)-trans-ACPD
Trans-(±)-ACP
(±)-trans-ACPD, un agonista de los receptores metabotrópicos, produce movilización de calcio y una corriente interna en neuronas de Purkinje cerebelosas cultivadas. -
GC11128
(±)-Vesamicol hydrochloride
(±)-AH5183 hydrochloride
(±)-clorhidrato de vesamicol ((±)-clorhidrato de AH5183) es un potente inhibidor del transporte vesicular de acetilcolina con una Ki de 2 nM. -
GC41685
(±)-WIN 55,212 (mesylate)
(±)-WIN 55,212-2 is a potent aminoalkylindole cannabinoid (CB) receptor agonist with a Ki value of 62.3 and 3.3 nM for human recombinant central cannabinoid (CB1) and peripheral cannabinoid (CB2) receptors, respectively.
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GC41213
(±)10-HDHA
10hydroxy Docosahexaenoic Acid, (±)10HDoHE
(±)10-HDHA is an autoxidation product of docosahexaenoic acid (DHA) in vitro.
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GC41214
(±)11-HDHA
11hydroxy Docosahexaenoic Acid, (±)11-HDoHE
(±)11-HDHA is an autoxidation product of docosahexaenoic acid (DHA) in vitro. -
GC40467
(±)11-HETE
(±)11-Hydroxyeicosatetraenoic Acid
(±)11-HETE is one of the six monohydroxy fatty acids produced by the non-enzymatic oxidation of arachidonic acid. -
GC40802
(±)12(13)-DiHOME
Isoleukotoxin diol
(±)12(13)-DiHOME is the diol form of (±)12(13)-EpOME, a cytochrome P450-derived epoxide of linoleic acid also known as isoleukotoxin.
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GC41191
(±)13(14)-EpDPA
(±)13,14-EDP, (±)13,14-EpDPE, (±)13,14-epoxy DPA, (±)13,14-epoxy Docosapentaenoic Acid
(±)13(14)-EpDPA (13,14-EpDPE) es el producto de la reacción de la epoxigenasa del citocromo P-450 con ácido docosahexaenoico (DHA). -
GC41192
(±)13-HDHA
13hydroxy Docosahexaenoic Acid, (±)13-HDoHE
(±)13-HDHA is an autoxidation product of docosahexaenoic acid (DHA) in vitro. -
GC41193
(±)14-HDHA
14hydroxy Docosahexaenoic Acid, (±)14-HDoHE
(±)14-HDHA is an autoxidation product of docosahexaenoic acid (DHA) in vitro. -
GC41194
(±)16(17)-EpDPA
(±)16,17 EDP, (±)16,17-epoxy Docosapentaenoic Acid, (±)16,17-epoxy DPA, (±)16,17-EpDPE
EDHF (endothelium-derived hyperpolarizing factor) is an unidentified mediator released from vascular endothelial cells in response to acetylcholine and bradykinin which is distinct from the NOS- (nitric oxide) and COX-derived (prostacyclin) vasodilators.
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GC41196
(±)16-HDHA
16hydroxy Docosahexaenoic Acid, (±)16-HDoHE
(±)16-HDHA is an autoxidation product of docosahexaenoic acid (DHA) in vitro. -
GC41197
(±)17-HDHA
17-hydroxy Docosahexaenoic Acid, 17-hydroxy DHA, (±)17-HDoHE
(±)17-HDHA is an autoxidation product of docosahexaenoic acid in vitro. -
GC41199
(±)19(20)-EpDPA
(±)19,20 EDP, (±)19,20-epoxy Docosapentaenoic Acid, (±)19,20-epoxy DPA, (±)19,20-EpDPE
EDHF (endothelium-derived hyperpolarizing factor) is an unidentified mediator released from vascular endothelial cells in response to acetylcholine and bradykinin which is distinct from the NOS- (nitric oxide) and COX-derived (prostacyclin) vasodilators. -
GC41202
(±)4-HDHA
4hydroxy Docosahexaenoic Acid, (±)4HDoHE
(±)4-HDHA is an autoxidation product of docosahexaenoic acid (DHA) in vitro. -
GC41203
(±)7(8)-EpDPA
(±)7,8-EDP, (±)7,8-EpDPE, (±)7,8-epoxy DPA, (±)7,8-epoxy Docosapentaenoic Acid
Docosahexaenoic acid is the most abundant ω-3 fatty acid in neural tissues, especially in the brain and retina. -
GC41204
(±)7-HDHA
7hydroxy Docosahexaenoic Acid, (±)7HDoHE
(±)7-HDHA is an autoxidation product of docosahexaenoic acid (DHA) in vitro.
-
GC41205
(±)8-HDHA
8hydroxy Docosahexaenoic Acid, (±)8HDoHE
(±)8-HDHA is an autoxidation product of docosahexaenoic acid (DHA) in vitro. -
GC33544
(±)-Methotrimeprazine (D6) (dl-Methotrimeprazine D6)
(±)-Methotrimeprazine-d6; dl-Methotrimeprazine-d6
(±)-Levomepromazina D6 ((±)-Metotrimeprazina D6) es la metotrimeprazina etiquetada con deuterio, que es un antagonista del receptor de dopamina D3 e histamina H1.
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GC31026
(±)-Tazifylline
(±)-Taziphylline es un antagonista del receptor H1 de histamina potente, selectivo y de acción prolongada.
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GN10155
(+)- Corydaline
(+)-Corydaline, D-Corydaline, NSC 406036
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GC13156
(+)-AJ 76 hydrochloride
Antagonista del receptor de dopamina