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(R)-PAD-PF2

Catalog No.GC80328 Copy One-Click Copy Product Info

(R)-PAD-PF2 is an isomer of PAD-PF2.

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(R)-PAD-PF2 Chemical Structure

Size Price Stock Qty
1mg
$252.00
In stock

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Sample solution is provided at 25 µL, 10mM.



Description of (R)-PAD-PF2

(R)-PAD-PF2 is an isomer of PAD-PF2. PAD-PF2 is a PAD family inhibitor, as well as a κ-opioid receptor agonist ( EC 50 = 7.55 μM) and an M1 muscarinic acetylcholine receptor antagonist ( IC50 = 12.3 μM).

Chemical Properties of (R)-PAD-PF2

Cas No. SDF
Formula C25H27Cl2N5O M.Wt 484.42
Solubility DMSO: 100 mg/mL (206.43 mM; ultrasonic and warming and heat to 60°C) Storage Store at -20°C
Shipping Condition Evaluation sample solution: shipped with blue ice. All other sizes available: with RT, or with Blue Ice upon request.

Complete Stock Solution Preparation Table of (R)-PAD-PF2

Prepare stock solution
1 mg 5 mg 10 mg
1 mM 2.0643 mL 10.3216 mL 20.6432 mL
5 mM 412.9 μL 2.0643 mL 4.1286 mL
10 mM 206.4 μL 1.0322 mL 2.0643 mL
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In vivo Formulation Calculator (Clear solution) of (R)-PAD-PF2

Step 1: Enter information below (Recommended: An additional animal making an allowance for loss during the experiment)

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Working concentration: mg/ml;

Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO ( Master liquid concentration mg/mL, Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug. )

Method for preparing in vivo formulation: Take μL DMSO master liquid, next addμL PEG300, mix and clarify, next addμL Tween 80, mix and clarify, next add μL saline, mix and clarify.

Method for preparing in vivo formulation: Take μL DMSO master liquid, next add μL Corn oil, mix and clarify.

Note: 1. Please make sure the liquid is clear before adding the next solvent.
2. Be sure to add the solvent(s) in order. You must ensure that the solution obtained, in the previous addition, is a clear solution before proceeding to add the next solvent. Physical methods such as vortex, ultrasound or hot water bath can be used to aid dissolving.
3. All of the above co-solvents are available for purchase on the GlpBio website.

Product Documents

Quality Control & SDS

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Average Rating: 5 ★★★★★ (Based on Reviews and 30 reference(s) in Google Scholar.)

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