Bliretrigine |
Catalog No.GC64658 |
Bliretrigine is a sodium channel blocker.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 1233229-75-8
Sample solution is provided at 25 µL, 10mM.
Bliretrigine is a sodium channel blocker. Bliretrigine has the effect of relieving pain[1][2][3].
[1]. WHO Drug Information, Vol. 35, No. 4, 2021. Geneva: World Health Organization; 2022.
[2]. Yoshihiro OYAMADA, et al. External medicinal preparation containing N2-{[1-ethyl-6-(4-methylphenoxy)-1H-benzimidazol-2-yl]methyl}-L-alanineamide for treating and/or preventing peripheral neuropathic pain. Patent AU2019306705.
[3]. Hironori Kinoshita, et al. Preparation of N2-[(benzimidazol-2-yl or imidazo[4,5-b]pyridin-2-yl)methyl]amino acid amide derivatives as inhibitors of sensory neuron specific sodium channel (SNS). Patent AU2009331179.
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