Fulvestrant 9-sulfone |
| Catalog No.GC49878 |
An estrogen receptor antagonist and a derivative of fulvestrant
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 98008-06-1
Sample solution is provided at 25 µL, 10mM.
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Fulvestrant 9-sulfone is an estrogen receptor antagonist and a derivative of the selective estrogen receptor degrader (SERD) fulvestrant .1 It binds to estrogen receptor α (ERα) and ERβ and inhibits estrogen-induced gene expression in a reporter assay in Ishikawa endometrial cells expressing an estrogen response element (ERE) reporter when used at concentrations ranging from 0.1 to 100 µM.
1.Nuttall, M.E., Pendrak, I., Emery, J.G., et al.Antagonism of oestrogen action in human breast and endometrial cells in vitro: Potential novel antitumour agentsCancer Chemother. Pharmacol.47(5)437-443(2001)
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